Ezempilo, Amalungiselelo
Isidakamizwa esithi "Claridol": imiyalo yokusetshenziswa, ukubuyekezwa
Ukuphefumula kwabantu kubantu kungabonakalisa ngezindlela ezahlukene. Kodwa kaningi ukucindezeleka kwesimiso sokuzivikela komzimba kuhambisane nezimpawu ezifana nobuhlungu emehlweni, imisipha, ukuvuvukala, impumulo egijimayo, ukukhwehlela nokunyakaza. Lezi zibonakaliso ziletha kabi kakhulu isiguli. Ngakho-ke, abantu abavame ukubhekana nezifo, ngokuvamile basebenzisa izidakamizwa ezinganciphisa ubunzima bezimpawu ezinjalo. Omunye wabo umuthi "Claridol". Imiyalo yokusetshenziswa, izithombe, izinkomba kanye nefomu lesidakamizwa kuhanjiswa ngezansi.
Incazelo yemithi, indlela yayo yokukhululwa, ukupakisha nokubunjwa
Luhlobo luni lokulungiswa okucutshungulwayo? Ngokusho kochwepheshe, lo muthi ungatholakala emafomu afana nalokhu:
- Amathebulethi "Claridol". Imiyalo yokusetshenziswa ibonisa ukuthi izidakamizwa zimhlophe, zizungezile, ziyizicabha, zihlanganiswe, futhi zikhona nomugqa wecala ohlangothini olulodwa.
Isithako esisebenzayo sale mithi i-loratadine. Ngaphezu kwalokho, lokhu kuhlanganiswa kuhlanganisa izingxenye ngendlela yama-silicon dioxide colloid, i-microcrystalline cellulose, i-starch, i-talcum ehlanzekile, i-methylparaben ye-sodium, i-magnesium stearate, amanzi ahlanzekile ne-sodium isitashi glycolate.
Ekuthengisweni kwalo mkhiqizo kufika amabhulashi kanye namabhokisi wekhadibhodi, ngokulandelana.
- Isiraphu "i-Claridol". Imfundo yokusetshenziswa ithi leli fomu lomuthi lenziwa ngesimo se-liquid elicwebe ebonakalayo enephunga elimnandi nelinambitheka elimnandi.
Isithako sayo esisebenzayo yi-loratadine. Futhi ekwakheni isiraphu kuhlanganisa i-sodium sucrose, i-propylparaben ye-sodium, i-citric acid, i-propylene glycol, isisombululo se-sorbitol, i-benzoate ye-sodium , i-sacdirin ye-sodium , i-disodium i-edetate, i-flavour yezithelo ezixutshwe, i-methylparaben, ilanga lokushona kwelanga, amanzi ahlanzekile ne-American ayisikhilimu.
Ungathenga le mithi ngamabhodlela weglasi elimnyama.
Isenzo somkhiqizo wokwelapha
Uyini umuthi "Claridol"? Imiyalo yokusetshenziswa, ukubuyekezwa kusikisela ukuthi lokhu kuyi-blocker ye-H1-histamine receptors, enomphumela wesikhathi eside. It kuvimbela ukuthuthukiswa kwemithi, futhi ikhulula i-leukotriene C4 ne-histamine kusuka kumangqamuzana amancane.
Umuntu akanakusiza ukusho ukuthi le mithi ine-antiexudative, antiallergic kanye ne-antipruritic imiphumela. Ivimbela ukuthuthukiswa kwe-edema yamathishu, inciphisa ukusikeka kwemisipha ebushelelezi futhi inciphise ukuguqulwa kwama-capillari.
Leli thuluzi alinamthelela kwisistimu ye-central central, imisebenzi ye-psychomotor, amakhono engqondo, ikhono lokusebenza nokunakekelwa, futhi akubangeli ubuthongo nokulutha, njengoba kungenangqondo ukungena kwi-BBB.
Izakhiwo eziphikisayo zokulwa nalesi sidakamizwa zithuthuka ngemva kwesigamu sehora bese zifinyelela ezingeni eliphezulu emva kwamahora angu-8-13 (ihlala usuku lonke).
AmaKinetics wemithi
Ingabe isidakamizwa se-Claridol sithatha? Imiyalelo yokusetshenziswa iqinisekisa ukuthi emva kokungenisa it is ngokugcwele futhi ngokushesha umxhwele kusukela digestive ipheshana. Ukudla ukudla kunciphisa inqubo yokuqoqa egazini ihora elilodwa lapho uthatha amaphilisi futhi akuthinteki ukumunca nganoma iyiphi indlela uma usebenzisa isiraphu.
Ukuhlangana kwezidakamizwa ezinamaprotheni e-plasma kungu-97.5%. I-metabolized isibindi ngokubunjwa kwe-derivative esebenzayo njenge-descarbonethoxyloratadine.
I-half-life ye-loratadine amahora angu-5 kuya ku-20 (ihlanganisiwe kanye nomchamo ne-bile).
Izimpawu zokusetshenziswa komuthi
Lapho isiguli sinikezwe umuthi "Claridol"? Imiyalo yokusetshenziswa (isiraphu namaphilisi anezinkomba ezifanayo) ithi le remedy iphumelela uma:
- I-pollinosis;
- Ukusabela okwenziwe okwenziwe nge-allergic kuya ukulunywa kwezinambuzane;
- Ukuvuselela unyaka wonke;
- Ukusabela kwe-pseudoallergic;
- I-rhinitis ye-allergen;
- Conjunctivitis ukugula;
- Ukunqunywa kwe-dermatoses yokuchithwa kwegazi;
- I-Urticaria (kubandakanya uhlobo olungapheli lwe-idiopathic yesifo);
- Ukuthakaza kwemvelaphi ehlukile;
- I-edema ka-Quincke.
Ukungafani kokuthatha lesi sidakamizwa
Kuziphi izimo akufanele usebenzise lesi sidakamizwa "Claridol"? Imiyalo yokusetshenziswa (izingane ezineminyaka engaphansi kweminyaka emibili le mithi ayimisiwe) ibonisa ukuphikisana okunjengokuthi:
- Ukukhulelwa;
- Hypersensitivity;
- Ukuncelisa.
Ngokunakekelwa okukhethekile, le mithi kufanele ikhuthazwe iziguli ezinezinkinga zesibindi (okubandakanya ukuhluleka kwesibindi).
Isidakamizwa esithi "Claridol": imiyalelo yokusetshenziswa
Yini eshiwo lo muthi, esichazwe ngenhla. Kufanele kuthathwe kanjani? Ngokusho kochwepheshe, lesi sidakamizwa sisetshenziswa ngomlomo kuphela.
Iziguli ezikhulile nezikhulile, kanye nezingane ezineminyaka engu-12 ubudala, imithi inqunywe u-10 mg kanye ngosuku.
Izingane ezineminyaka engu-2-12 ezinesisindo somzimba ezingaphansi kuka-30 kg zinconywa ukuba zithathe ama-5 mg wezidakamizwa kanye ngosuku.
Ngokuqondene nezingane ezineminyaka engu-2-12 enesisindo somzimba esingaphezu kuka-30 kg, banikwa 10 mg wemithi kanye.
Akunconywa ukubeka lo muthi kubantwana abangaphansi kweminyaka emibili ubudala.
Abantu abanesifo esibindile somzimba banqunywe esilinganisweni sokuqala esilingana no-5 mg ngosuku.
Imiphumela emibi emva kokuthatha imithi
Isidakamizwa sikaClaridol sikhuthazwe kanjani iziguli? Imfundo yokusetshenziswa ithi ukusetshenziswa kwalesi mithi kungabangela ukusabela okulandelayo:
- Izinsizwa, ukuhlanza, isizungu, ukungasebenzi kwesibindi, ukulala;
- Ukukhathala okwandisa, ukuphazamiseka, i-tachycardia;
- Isikhumba, ukusabela okweqile (kufaka phakathi i-rash ne-anaphylaxis), i-alopecia;
- Umlomo omile, ukuzwakalisa, ukucabangela, ukuzithemba, isisu somzimba.
Ukusebenzisana kwezidakamizwa
Uma isidakamizwa esinikeziwe sihlangene ne-cimetidine, ketoconazole, noma i-erythromycin, ukwanda kokuhlushwa kwezinto ezisebenzayo egazini kungenzeka, okungenayo umphumela ku-ECG futhi kungabi nokubaluleka komtholampilo.
Ama-inducer anjalo , njenge-barbiturates, i-phenytoin, i-rifampicin, i-zixorin, i-tricyclic anti-depressants, i-phenylbutazone, ne-ethanol, ukunciphisa ukusebenza kwe-loratadine.
Ukubuyekezwa kwesineke
Abathengi bathi izidakamizwa "i-Claridol" iyinhlangano yokulwa ne-antiallergic esebenzayo. Iqeda masinyane izimpawu ezinjengezinkomba ezifana nokukhipha, ukukhwehlela, ukukhwehlela nabanye, okubangela ekuthuthukiseni isimo sesiguli.
Ukungaphumeleli kwalesi sidakamizwa kubandakanya ukutholakala kwemiphumela emibi eminingi, kanye nokungabi nethuba lokunikeza abesifazane abakhulelwe nabamama ababelethayo.
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