Imithi yokwelashwa
Izidakamizwa "i-Bloktran" imiyalelo yokusetshenziswa njenge-agent e-antihypertensive, okuyinto ephikisanayo nama-receptors akhethekile we-angiotensin II. Ukusetshenziswa kwalesi sidakamizwa kunganciphisa ingcindezi emjikelezweni omncane wegazi, ukunciphisa ukumelana kwemithambo yegazi, izinga le-aldosterone ne-adrenaline. Ngaphezu kwalokho, lesi sidakamizwa "iBloktran", imfundo lapho uhlelo lokusebenza luhlale luhlanganiswe khona, ngokuyimpumelelo kuvimbela ukuthuthukiswa kwe-hypertrophy ye- myocardial, inomthelela wokuba nesifo esibucayi futhi ikhulise ukubekezelelana komthwalo. Lokhu okubaluleke kakhulu kubantu abahlukunyezwa yinhliziyo. Ngokuqondene nezici ezikhethekile ze-pharmacokinetics yalesi sidakamizwa esinamandla, ama-plasma aphezulu kakhulu agcinwa ngemva kwamahora ayisihlanu kuya kwangu-8 emva kokusetshenziswa. Umthelela omkhulu wokwelapha utholakala ngemuva kwamasonto amathathu kuya kwayisikhombisa wemithi ejwayelekile "iBoktran", intengo yayo ehluka kusuka kuma-ruble angamakhulu amathathu kuya kwangu-4.
Incazelo yokubunjwa kwemithi
Lesi sidakamizwa esinamandla kakhulu sakhiwa ngesimo samathebulethi azungeze umbala ophuzi obomvu. Njengento esebenzayo ekubunjweni kwe-dragee ama-milligram angu-50 we-potassium losartan. Izithako ezengeziwe ziyi-starch, i- microcrystalline cellulose, i- lactose, i-silicon dioxide, i-magnesium stearate ne-povidone. Ukwakhiwa kwegobolondo kuhlanganisa izinto ezifana ne-talcum, i-hypromellose, i-yellow-orange sycovitis ne-polysorbate-80. Ngaphezu kwalokho, inani elincane le- titanium dioxide ne-copovidone.
Izinkomba zokusetshenziswa
Thatha iphilisi "imfundiso yeBloktran" yokusetshenziswa iluleke ukwelashwa kwesifo somfutho wegazi ophezulu. Ngaphezu kwalokho, le nsizakalo ibhalwe ngokuqinile ukuze ilaphe iziguli ezinokukhubazeka kwenhliziyo okungapheli.
Uhlu lwama-contraindications wezokwelapha
Qala ukwamukelwa kwezidakamizwa "imiyalo yeBloktran" ukuze usebenzise ngokuqinile ukuthi awuncoma uma kwenzeka ukuphelelwa amanzi, ukuphefumula kwegazi kanye ne-hypotension. Ubudala bezingane, i-lactation kanye nesikhathi sokukhulelwa zifakiwe kuhlu lwamacala okuqinela. Ngaphezu kwalokho, ngokuyinhloko akudingekile ukuthi uthathe lawa amaphilisi uma kwenzeka i-hypersensitivity i-losartan potassium noma ezinye izici. Ngokunakekelwa kahle, lesi sidakamizwa esinamandla kakhulu kufanele sisetshenziswe ekunakekeleni kwe-renal nokuqina okukhulu kwe-hepatic.
Uhlu lwemiphumela emibi
Ukusetshenziswa okuqhubekayo kwamathebulethi "e-Bloktran" kungabangela izinwele, i-asthenia, ukuleleka, isizungu, nobuhlungu besisu. Kungase kube ne-gastritis, isifo sohudo, isicanucanu nokuhlanza. Kungase kube nokungqubuzana komzimba, ukuxubana, ukuphazamiseka kokulala, i-ataxia, i-hypostases, ukunambitheka okungahambi kahle, ukukhala ezindlebeni, ukuthuthumela, ukuguqulwa kwe-paresthesia kanye ne-peripheral neuropathy. Ukoma, sinusitis, i-myalgia, i-syncope, i-conjunctivitis ne-rhinitis - konke lokhu kuyimbangela yokusetshenziswa isikhathi eside kwesidakamizwa. I-Dispno, i-bronchitis, i-migraine, umlomo omile, i-anemia, i-angina ne-bradycardia nayo ingathuthuka ngenxa yokusebenzisa lesi sidakamizwa "i-Bloktran". Lo muthi ungavusa ama-angioedema, ama-hives, i-hyperkalemia, ukwehluleka kwe-libido ne-alopecia.