ImpiloAmalungiselelo

"Flosteron": ukubuyekezwa. "Flosteron" ngoba komzimba

Bewazi yini ukuthi lena izidakamizwa ngokuthi "Flosteron"? ochwepheshe lezivakashi bathi kuba ithuluzi jikelele engasetshenziswa ezimweni ezihlukahlukene sokugembula.

Ngalokho izakhiwo wathi ifomu izidakamizwa lapho kungenzeka ukuthola futhi indlela yokusebenzisa, kuzoxoxwa ngakho esihlokweni ethulwa.

Okufakiwe, ukwakheka kanye ngesimo

izidakamizwa "Flosteron" Lapho ithengiswe? Izibuyekezo zabantu abaye babike ukuthi imithi angathengwa ngasiphi ekhemisi. Futhi, ezinye iziguli ziye walithenga-intanethi.

Ithuluzi linaso izingxenye esebenzayo njengoba betamethasone disodium phosphate futhi betamethasone dipropionate. Ngaphezu kwalokho, ukwakheka kufaka nomuthi asekelayo izakhi ngesimo sodium chloride, i-sodium carmellose, polysorbate 80, i-sodium edetate, methyl paraben, Gcoba i-Benzyl utshwala, hydrochloric acid bagxila, propylparaben, i-sodium ne-hydrogen phosphate dihydrate, polyethylene glycol namanzi ahlanzekile.

Medicine "Flosteron" okuyinto izilinganiso ezibekwe, ukukhiqiza ukumiswa for umjovo. Itholakala ampoule (1 ml) e uhlaka amaphakheji.

pharmacodynamics

Kanjani lesi sidakamizwa "Flosteron"? Yokusetshenziswa (imibono kusukela ochwepheshe ngalokhu ithuluzi kukhona uhlamvu omuhle kuphela) lithi eselaphayo izidakamizwa okukhulunywe ngabo lapha bangabantu ama (ie, esikhundleni zokwenziwa hormone adrenal). They possess izakhiwo immunosuppressive, anti-rheumatism futhi eqeda ukuvuvukala.

Betamethasone nomthelela homeostasis glucose, amandla umzimba izidakamizwa kanye ne-hormone okuthiwa yokudla okunempilo kusukela pituitary anterior.

Kuze kube manje, isimiso isinyathelo of glucocorticoids bengayiqondi ngokugcwele. Nokho, kukhona umbono wokuthi inqubo yenziwa umthelela wabo ku emangqamuzaneni. Ochwepheshe bakholelwa ukuthi cytoplasm yengqamuzana, zikhona izinhlelo ezimbili yokwamukela, futhi betamethasone kunomthelela oqonde ngqo iqhaza ekhethekile GCS receptor. Ngakwelinye ihlangothi, ama-receptor mineralocorticoid neqhaza ukulawulwa-sodium potassium umzimba namanzi futhi electrolyte ibhalansi.

Ngama-corticosteroid ngokuthi izinto fat-encibilikayo. Bona kalula ukungena ngokusebenzisa ulwelwesi cell esitokisini target.

Ngakho, empeleni sisuke sicabanga izidakamizwa esekelwe izinqubo ezithile kwamakhemikhali kwenzeka ezingeni yamangqamuzana ezinto eziphilayo.

Pharmacokinetics

Betamethasone dipropionate amuncwa umzimba kancane, kodwa inikeza umphumela sasivumela eside. Kuye mode yokuphathwa kungaba sifinyelele nomphumela jikelele noma wendawo.

Ubuningi esiphezulu izidakamizwa waphawula ngemva naphakathi-articular ekuphathweni emva kwemizuzu engu-30. Umuthi plasma ngokushesha amaprotheni ngokwanele nakanjani. It kalula lingena izithiyo igazi-izicubu, kuhlanganise esinomhlapho.

Izidakamizwa umzimba esibindini ukuze metabolites esingasebenzi. Bheke zezinto asebenzayo kwenzeka izinso, futhi kanye Bile futhi ubisi kancane webele.

ubufakazi

imijovo Uma iziguli okunqunyiwe "Flosteron"? Uphenyo odokotela bathi umuthi jikelele engasetshenziswa ukwelapha izifo ezehlukene. Ngokusho imiyalelo, umuthi isetshenziselwa:

  • ubuchopho edema;
  • igazi, kuyashaqisa, ukusha, anaphylactic, ukusebenza, cardiogenic futhi ezinobuthi uthuthumele;
  • izifo yemvelo letindzala sezicubu zezinzwa (isib lupus erythematosus, usizi thyrotoxic, ikhoma hepatic, i-rheumatoid arthritis);
  • isifuba somoya bronchial ezinzima;
  • ukusabela anaphylactoid ;
  • ukuvimbela ukuvuvukala kanye nezibazi ngemva kokungenwa uketshezi caustic.

Ngingakwazi ukusebenzisa "Flosteron" ngoba komzimba? Izibuyekezo ochwepheshe ukubika ukuthi lokhu izidakamizwa siyasebenza kakhulu kuzibonakalisa ukusabela imvelo nomzimba. Ngakho-ke, ngokuvamile ezinqunyiwe:

  • isifuba somoya bronchial, esingalapheki noma rhinitis ezithile zonyaka;
  • psoriasis, atopic dermatitis kanye contact keloids;
  • kollagenozah;
  • Extra articular rheumatism, sokuqaqanjelwa yiqolo, umfutho tenosynovitis, myositis, synovitis, i-osteoarthritis posttraumatic, epicondylitis, cystic;
  • ukulunywa yizinambuzane;
  • yiluphi uhlobo komzimba nezinto;
  • izilonda emathunjini.

Izimo

Lapho hhayi ukusebenzisa izidakamizwa "Flosteron" (imfundo, ke libuyekeza nomuthi izokwethulwa kamuva)? It is hhayi ezinqunyiwe:

  • kwamathambo, isilonda esiswini, isifo sofuba diverkulite, ukufiphala;
  • syndrome, Cushing, thrombophlebitis, izifo sibi viral, webhaktheriya noma fungal, isifo sikashukela;
  • imisebenzi enzima futhi ezibuhlungu, ngaphambi nangemva lokugoma (amasonto amabili);
  • idiopathic purpura thrombocytopenic (esicutshini);
  • ukungabi khona ukuvuvukala emalungwini;
  • uhlobo ithambo nokubhujiswa ngokuhlanganyela, ukungazinzi ngokwezomnotho ngokuhlanganyela;
  • azalwa naso noma ukopha okubangelwa ngokuthatha anticoagulants;
  • lactating abesifazane, izingane ezingaphansi kweminyaka emithathu yozwela anda.

Nomuthi "Flosteron": yokusetshenziswa

Nobufakazi mayelana izidakamizwa abasakwazi edidayo.

Kanjani lokhu izidakamizwa kumele kusetshenziswe?

Ukuze kuthinte nesineke systemically, nomuthi iqondiswa intramuscularly. Imijovo eyenziwe gluteal kwemisipha (ezijulile) ka 0.1-0.2 ml njalo emavikini 2-4.

Njengoba okunqunyiwe "Flosteron" ngoba komzimba? ochwepheshe lezivakashi bathi umuthi onjalo ngokuvamile sisetshenziswa uma kwenzeka acute komzimba uhlamvu. Kulokhu, umjovo nayo wenza intramuscularly ku isamba 1.2 ml (umthamo owodwa).

Lapho isicelo ihlelwe ngokulandelana kwezihloko, umthamo we izidakamizwa ingahluka kakhulu. Ngokuvamile, it kufana ml 0.25-2.

Ngo-psoriasis, dermatitis atopic, eczema nezinye izifo zesikhumba imithi intradermally phambili.

Uma kudingeka, ekwakhiweni ngicele impumuzo ubuhlungu kungenziwa exutshwe procaine noma lidocaine.

Izingane 3-5 iminyaka umthamo kokuqala umuthi 0.3 ml futhi izingane eminyakeni 6-12 ubudala - 0.6 ml.

Izidakamizwa "Flosteron": Izibuyekezo

Ehlaziya ukusabela lezazi sikhungo abakhona, singaphetha kahle ukuthi izidakamizwa siyasebenza kakhulu. Ngokusho imibiko yodokotela, lokhu imithi isetshenziswa izifo kabi ebuchosheni ngempela, ezicutshini, ukusabela anaphylactoid, nokunye. D.

Njengoba for iziguli, abayivezi ngaso sonke isikhathi ukushiya okubuyayo mayelana nokumiswa "Flosteron". Izibuyekezo zabantu bathi lo muthi ngokuvamile kakhulu kubangela engemihle. Lezi zihlanganisa isiyezi, ukucobeka thinning kwesikhumba, isisindo somzimba kanye ngaphezulu.

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