"Pyrazinamide" Tablets babe amagciwane noma umphumela bacteriostatic anti kuncike okuhlushwa. umsebenzi izidakamizwa inakekelwa kuphela ngaphansi kwezimo esidi (ngesikhathi pH 5.6 kanye ngezansi). ku inhlabathi imithi kungenzeka ukuthuthukiswa ukumelana, okuyinto kunciphisa amathuba usebenzisa imithi nezinye ejenti antitubercular. Ukulungiselela "Pyrazinamide" (incwadi yeziyalezo kuqinisekisa lokhu) ndlela iphumelela kakhulu lapho sofuba elimazayo njengoba wathola okokuqala, icubungula caseous-nenyumoniya uhlobo tuberkulomah, lymphadenitis caseous. Umuthi kwehlisa zokuthutha izindleko urate futhi uric acid, Hyperglycemia kungabangela. Umuthi kusukela pheshana emathunjini cishe ngokuphelele neqondakala ngokushesha. Plasma amaprotheni uxhumano nomsebenzisi nomuthi 10-20%. Ngemva kwehora noma amabili kukhona emakamu esiphezulu izimali. Imithi is kahle okuye kwasakazwa eminyakeni uketshezi lomzimba nezicubu, kufanele zibekwe izitho, kuhlanganise emaphashini, isibindi, izinso kanye nezinye izingxenye zesifunda encapsulated izilonda tuberculous. Kusho uphasisa Bbb. Umzimba kwenzeka esibindini.
ubufakazi
Nomuthi "pyrazinamide" (izimpendulo wezazi siliqinisekise) kuyisinqumo esingcono lokuqala ekwelapheni isifo sofuba.
Umthamo lwemithi
Kwatholakala ukuthi monotherapy akuyona ngempumelelo ngokwanele. Mayelana leli bhukwana izidakamizwa "pyrazinamide" imfundo uncoma ukusetshenziswa lihambisana namanye nemithi abane-TB ephilayo. Kubantu abadala, umthamo kuyinto 30-35 mg / kg kanye ngosuku. Ezigulini enesisindo esingaba amakhilogremu esingaphansi amahlanu, umthamo kuyinto amaphilisi amathathu (1.5 g). Lapho mass ingaphezu 50 kg kufanele baphuze amaphilisi 4. (2 g). Ezinganeni umthamo esiphezulu - 2 amagremu. Umuthi esithathwayo ngokudla. Kunconywa ukuthi uphuze imithi ngesikhathi sasekuseni.
"Pyrazinamide" lisho ukuthini. Yokusetshenziswa. Izixwayiso
Imithi ukweqisa izidakamizwa kuhambisana oda kadokotela azibangelwa. Uma uthola semali zomuthi waphawula imiphumela emibi isimiso sezinzwa esiyinhloko - isiyezi, ubuhlungu bekhanda kanye nabanye. amanothi disorder esibindini, kungenzeka dyspepsia. Uma ushevu kuboniswe ukwelashwa lingaze. Ngaphambi naphakathi ukwelashwa kwe-TB ezigulini engaphezu kuka-60 Kwenziwa ukuqapha yenyanga izinkomba bilirubin, AST, acid uric no-ALT. Ngo iziyaluyalu kwesibindi kudinga ukususwa zomuthi. Ngo iziguli sikashukela maningi amathuba ukuthuthukisa kahle kungakhuphula izinga likashukela. Lapho kuhlangene imithi ukuthatha imithi "rifampicin" kungabonakala nasemkhakheni hepatotoxicity. Lapho kuhlanganiswe ukulungiselela isicelo "Probenecid" Cishe wehlise excretion futhi ngenxa yalokho, anda ubuthi. Kungase kube cross-ukuzwela ngemithi "INH", "Ethionamide" nicotinic acid nezinye izindlela kokuba efanayo amakhemikhali isakhiwo. "Pyrazinamide" imithi (yokusetshenziswa kuqinisekisa lokhu) ezifaneleke iminyaka emihlanu. Ukwakheka lilondolozwe emaphaketheni esivaliwe, ezindaweni bavikelekile ukukhanya.