Kusho "simvastatin" umyalelo ku isicelo lichaza izidakamizwa njengoba hypolipidemic kungokwalabo iqembu, futhi ama-statin kukhona inhibitors ka HMG-reductase uhlobo CoA. Lokhu nomuthi kuyinto prodrug, kusukela oyiyo elikhona avaliwe, okuthiwa lactone indandatho okuyinto, ngemva kokufaka umzimba womuntu hydrolyzed. Umuthi 'Simvastatin "(Ukufundiswa on isicelo yalesi kugxila) kusiza ukunciphisa amazinga igazi triglyceride futhi Esilula cholesterol Imininingwane. Ngesikhathi esifanayo ukuthuthukisa nomphumela oqabulayo luqala ngemva angathi ishumi nambili bebonke noma nane kusukela kuqale ukusetshenziswa, futhi umphumela esiphezulu kufinyelelwa yesine neviki lesithupha.
Umuthi senziwa ikakhulukazi ngesimo amaphilisi round biconvex. Ukwakheka pellet ngamunye isithako esebenzayo main has angu amabili simvastatin. izingxenye engeziwe lactose, polyvinylpyrrolidone, i-calcium stearate, citric acid, hypromellose, microcrystalline cellulose, hydroxyanisole butylated, ascorbic acid, corn isitashi, ama-titanium dioxide, talc futhi Macrogol 4000.
Linqume lipid-ukwehlisa izidakamizwa "Simvastatin" imfundo manual weluleka, isibonelo, ukuze kwelashwe abantu abaphethwe hypercholesterolemia eyinhloko. Nokho, ukusebenzisa ithuluzi kulesi simo kubalulekile kuphela uma ukudla okungenamsoco. "Simvastatin" izidakamizwa nakho excellently ukuhanjwa ekwelapheni hypercholesterolemia kuhlanganiswe. Izinkomba kanye zihlanganisa izifo ezifana hypertriglyceridemia.
Thatha lezi amaphilisi akuvunyelwe nakancane kubantu abaphethwe amafomu okunzima iziyaluyalu kwesibindi kanye ezinzima esingamahlalakhona kwezinso. Uma hypersensitive ukuba simvastatin noma iziphi izakhi asizayo ochwepheshe efanayo ukuncoma ayeke ukuthatha lipid-ukwehlisa izidakamizwa "Simvastatin". Yokusetshenziswa akufanele ukwabela izidakamizwa iziguli azifinyelelanga iminyaka eyishumi nesishiyagalombili ubudala, abesifazane abakhulelwe omama abasebasha ibele. Ngokunakekela okukhulu kumele usebenzise lezi amaphilisi iziguli isifo sesibindi, hypotension noma isithuthwane. Ngo ukuluthwa utshwala chronic ezinzima isifo sezinso ukuthatha imithi "Simvastatin" kufanele kuphela ngaphansi kweso lwezokwelapha. Ngaphezu kwalokho, uhlu Izimo isihlobo zibandakanya anda futhi kwehle lwamathambo imisipha ithoni.
Kuze kufike imiphumela engemihle engase cuphuluza izidakamizwa eyanele "Simvastatin", into yokuqala lapha kuyadingeka ukwaba ingozi pancreatitis, peripheral neuropathy, hypotension, myopathy, volchanochnopodobnogo syndrome, rhabdomyolysis futhi thrombocytopenia. Ngaphezu kwalokho, ukuquleka kungenzeka, isiyezi, ukubuyisa, ukungakuthandi ukudla, angioedema, amawala, siwasebenzise, urticaria, eosinophilia, photosensitivity, vasculitis, imfiva, imisipha paresthesia, Alopecia, futhi igazi.