Impilo, Amalungiselelo
"Levocetirizine": yokusetshenziswa, incazelo izidakamizwa, analogue kanye nokubuyekeza
Kungakanani buyisidakamizwa "levocetirizine"? Intengo yaleli izidakamizwa izokwethulwa ekupheleni. Uyofunda indlela ukusebenzisa izidakamizwa, kusho ukuthi ukhulunyelwa 'kodokotela kanye neziguli, ifomu kuwo ikhangiswa iphinde lokho izakhiwo.
Ifomu kanye nokusungulwa izidakamizwa emaphaketheni
Ukulungiselela "Levocetirizine Teva" ikhishwe ngendlela amaphilisi. nempahla yabo esebenzayo levocetirizine dihydrochloride. Futhi izidakamizwa yizici ezincane ngesimo monohydrate lactose, microcrystalline cellulose, magnesium stearate futhi Silica colloidal.
Thenga le nomuthi kungaba amakhadibhodi amabhokisi, okuyinto ezibekwe aluminium amabhamuza ukuze 7, 14 noma 10 amaphilisi.
pharmacodynamics zomuthi
Yiziphi amaphilisi "levocetirizine"? Yokusetshenziswa uthi nempahla yabo esebenzayo isomer levorotatory ka cetirizine, okuyinto ethatha njengoba omelene kakhulu sokukhohlwa elinamandla neuropathy H1-yokwamukela.
izidakamizwa Okubukwe kungathinta gistaminozavisimuyu isigaba komzimba nezinto, ukunciphisa yokufuduka eosinophils, wehlise semithambo permeability kanye ukukhululwa kwe balamuli ukuvuvukala.
Lokhu kuvimbela hhayi kuphela ukuthuthukiswa nomuthi kodwa futhi attenuates ukuvuza komzimba. It has izakhiwo antipruritic anti-exudative futhi has anticholinergic okuncane kanye antiserotoninovoe umthelela. Ngesikhathi Kunconywa ngemithamo zokwelapha zalesi izidakamizwa cishe akakubangeli ukozela kanye ukucobeka.
Pharmacokinetics
Yini imingcele kinetic babe "levocetirizine" ithebhulethi? Yokusetshenziswa ubika ukuthi ngemva umthamo owodwa we imithi ngempumelelo zayo zokwelapha e-50% eziguli waphawula emva kwemizuzu 12-13 futhi 95% eziguli - emva kwemizuzu engaba ngu-60 (umphumela uyaqhubeka ngesikhathi ezinsukwini ezalandela).
Lokhu nomuthi has pharmacokinetics komugqa. Uma ukungenisa it is ngokushesha ugxile kungakhathaliseki ukudla.
I bioavailability zomuthi ifinyelela ku-100%. I lokuhlushwa eliphezulu kakhulu ejenti asebenzayo waphawula emva kwemizuzu 55 emva kokungenisa, namaprotheni ngibopha cishe 90%.
Izidakamizwa umzimba kwenzeka esibindini futhi excreted ngu izinso ewonke.
izinkomba
"Levocetirizine" Tablets kuboniswa ngoba impatho siyefana lezi zifo ezilandelayo:
- pollinosis (noma okuthiwa hay fever);
- rhinitis futhi conjunctivitis Lokudabuka nomzimba, ephelezelwa ukulunywa, lacrimation, rhinorrhea, sneezing, futhi ububomvu we conjunctiva;
- angioedema;
- urticaria, kuhlanganise idiopathic, okuyinto agelezela ifomu ezingamahlalakhona;
- dermatosis nomzimba, izimpawu ukulunywa nesimungumungwane.
Izimo
Hlobo luni Izimo kufanele wazi ngaphambi kokusebenzisa "levocetirizine" ithebhulethi? Yokusetshenziswa Ngokusho la enqabela, njenge:
- yobudala ingane cishe iminyaka engaba yisithupha;
- CRF ibe mibi kakhulu njengenkemba,
- ngesikhathi sokukhulelwa;
- hypersensitivity izidakamizwa izakhi, futhi eqaphela ukuthi piperazine nemikhiqizo yalo;
- ngesikhathi sokuncelisa ibele.
Ngokunakekela okukhulu nomuthi ezinqunyiwe CRF kobukhulu okuncane noma okusesilinganisweni amafomu, kanye nokuguga (ngenxa ukuncipha kungenzeka e filtration glomerular).
Izidakamizwa "levocetirizine": yokusetshenziswa
Ngokwe-art, nomuthi asebenzayo ekuphathweni temlomo, kungakhathaliseki ukuthi ukudliwa kokudla. Izibhebhe okufanele zithathwe ngamanzi plain.
Izingane abaneminyaka engama eziyisithupha, kanye neziguli omdala Kunconywa umthamo yesikhathi esisodwa 5 mg. Lona umthamo esiphezulu ngelanga.
Isikhathi isilinganiso kwelashwa amasonto 3-6, kuye ngobucayi izimpawu. Ngo Ukuchayeka isikhashana ukwelashwa allergen kungaqedwa esikhathini esingaphansi kwesonto.
Njengoba kwezimo ezimbi kakhulu ezingalapheki, iguliswa, bangase okudinga izidakamizwa izinyanga eziyisithupha.
iziguli ezindala labo isifo sesibindi akudingeki ulungise umthamo.
Lapho umthamo isifo sezinso kufanele kushintshwe ngokuvumelana QC nesineke:
- engaphansi kuka-10 ml ngomzuzu - kokuthola imithi contraindicated;
- engaphansi kuka-30 ml ngomzuzu - 5 mg izinsuku 6;
- 30-49 ml ngomzuzu - 5 mg izinsuku 4;
- ezingaphezu kuka-50 ml ngomzuzu - 5 mg izinsuku 2.
ukusabela ezingezinhle
Iziphi izinkinga zokwelashwa kungenzeka ngenkathi ephethe izibhebhe "levocetirizine"? ochwepheshe lezivakashi uthi ukusabela elandelayo enqabayo:
- ukukhathala, ukuphathwa ikhanda, isiyezi, ukucasuka;
- ukozela, angaboni kahle, ubuhlungu besisu, ikhanda;
- lokujabulela ukoma emlonyeni, dyspepsia, dyspnea, ukukhathala;
- isicanucanu, isisindo somzimba, tachycardia;
- komzimba ezifana angioedema, awahlabi esikhumbeni, ukulunywa, urticaria.
Izimpawu ukweqisa izidakamizwa
Lapho ethola iphilisi ezingaphezu kwesisodwa ngosuku iziguli omdala ukuthuthukisa ukozela, nezingane - injabulo nokukhathazeka.
Therapy ye kwezimo ezinjalo kuyehla kube impatho lingaze nge esiswini lavage futhi engayitholi sorbents.
izidakamizwa ekuhlanganyeleni
Kanyekanye reception "levocetirizine" nge "theophylline" umthamo 400 mg, kunciphisa imvume ingqikithi ngowokuqala 16%, kodwa akazange siguqula kinetics lakamuva.
Ngo abantu ebucayi babambisane nokuphathwa izidakamizwa nama ejenti ethu ukuthi zivimbela isimiso sezinzwa esiyinhloko, kuhlanganise i-ethanol, kungase potentiate imiphumela Ukuncipha.
Synonyms, analogs, futhi izindleko zomuthi
Uyini izidakamizwa analogue "levocetirizine"? Amaconsi kwezokuphatha temlomo kungaba nomphumela ofanayo njengoba ifomu tablet. Ngakho-ke, abanye ochwepheshe batusa esikhundleni kubhekwe izidakamizwa izindlela ezifana "Pollezin" futhi "Suprastineks" (amathonsi). Ngaphezu kwalokho, analogs yalesi izidakamizwa kukhona "Allertsetin ',' Zestril ',' Alerza", "Rolinoz", "Zirtek", "Zintset", "Tsetrin", "Allertek", "Zetrinal", "Amertil" "cetirizine" "Zodak", "Letizen S", "Parlazin".
Ngokuqondene omqondofana ke izidakamizwa ezinjalo zihlanganisa lezi ezilandelayo: "Zodak" Allerset-L "," Zenaro "," levocetirizine "Sandoz", "Tsetrilev", "ka-L CET", "Tsezera", "Glentset", "Suprastineks" "Aleron" Express "," Ksizal ".
Ingakanani le izidakamizwa ngokuthi "levocetirizine"? wentengo uyahluka ruble 170-290.
nobufakazi
Iningi izibuyekezo mayelana izidakamizwa "Levocetirizine-Teva" akhayo. Iziguli eziningi ohlale uhlushwa ukusabela okuhlukahlukene umzimba uxabane nawo, ngokuvamile kakhulu ukusebenzisa lolu izidakamizwa. Bathi "levocetirizine" buyindlela ephumelelayo hhayi kuphela ukulapha eside, kodwa futhi ngoba usizo lokuqala uma umzimba wakho uxabana ne yesizini, noma unyaka wonke. Lokhu ukulungiselela ikuvumela ukuba alondoloze impilo ezingeni elifanele, ekuqedeni zonke izimpawu ezingemnandi bemvelo nomzimba.
Phakathi Izibuyekezo ezingezinhle ungathola lezo sithi izidakamizwa kubangela ukozela, ukukhathala ukucasuka. Odokotela bathi lapho ithola umthamo efanele kwezidakamizwa ukusabela ashiwo ezingavamile kakhulu.
"Levocetirizine" noma "Cetirizine": okuyinto engcono?
Lo mbuzo wabuzwa iziguli eziningi ohlale uhlushwa komzimba. Ochwepheshe ukubika ukuthi ezimbili wethule izidakamizwa yokubhekana ngokuphumelela kulo msebenzi. Kodwa, njengoba umkhuba imibukiso, "levocetirizine" ikhava tablet futhi aqede inqwaba izimpawu nomzimba.
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