ImpiloAmalungiselelo

Yokusetshenziswa "Zolpidem". Izibuyekezo futhi analogue

Uyini izidakamizwa "Zolpidem"? Yokusetshenziswa, omqondofana nokubonakaliswa lokhu izidakamizwa sizobuye kubhekwe.

Ukuma kanye nokwakheka

Equkethe izidakamizwa "Zolpidem"? Umhlahlandlela uthi nomuthi kubhekwe siqukethe izinto asebenzayo, njengabo zolpidem hemitartrate (10 mg), kanye nesimo sezulu asekelayo. Itholakala amaphilisi elimhlophe okuyizinto ezingenawo ezibekwe Valium amaphakheji planimetric yizicucu 15.

izici kwemithi

Kanjani izidakamizwa ehilelekile? Elikushoyo ngakho yokusetshenziswa? "Zolpidem" isimiso yayo wokusebenza kuyafana benzodiazepines. nomuthi Active uyakwazi bembonisa okuyiluthayo, anticonvulsant, amnesic, anxiolytic futhi izakhiwo sine.

I asebenzayo nemithi isici liyithinta ngokuqondile kwi-receptor benzodiazepine lokuqala nezinhlobo yesibili. Lokho kwenza kuvulwa iziteshi anionic neuronal usebenzisa la mangqamuzana Gaba ukuthi kamuva kuholela zamanje anda chlorine.

Ukuxhumana zomuthi kwenzeka ngokukhetha. Kule ndaba, umphumela izidakamizwa kuncike umthamo. Ngakho, imithamo ephansi avunyelwe ukufinyelela amnestic, miorelaksiruyuschee futhi izakhiwo anxiolytic futhi ukuvimbela umphumela okuyiluthayo

Kuyini ephawulekayo lokhu imithi? Elikushoyo ngakho yokusetshenziswa? "Zolpidem" ubuthongo esheshisa inqubo futhi kuthuthukisa nobuthongo. Kufanele kuphawulwe ukuthi ngemva kokuvusa ukozela e isiguli ingagciniwe.

izakhiwo kinetic

kanjani ukumuncwa lesi sidakamizwa "Zolpidem"? Ukusetshenziswa kwalesi imithi, noma kunalokho Isikali kwawo kuxhomeke kulokho ubufakazi. Ngemva kwemizuzu engaba ngu 30-110 esebenzayo izidakamizwa izidakamizwa ifinyelela izinga esiphezulu egazini. He cishe zonke nakanjani plasma amaprotheni bioavailability salo 70%.

Phezu kokuthola nomuthi e nezicubu isibindi othola ukusabela umzimba, okuholela kwetinhlavu nemikhiqizo esingasebenzi. Ziyakwazi ezinye ekhombisa umchamo futhi mayelana 40% - ne indle.

Isikhathi isigamu-ukuphila umuthi imizuzu 150. Lapho nokwephula kwesibindi, le nqubo enwetshiwe emahoreni angu-10.

Izidakamizwa "Zolpidem" imfundo on isicelo, isithombe zazo kukhonjisiwe ngezansi, ingena obisini lukamama.

Ukuze lokho ezinqunyiwe?

Yibuphi ubufakazi kubhekwa umuthi? Elikushoyo ngakho yokusetshenziswa? "Zolpidem" - i-tablet senzelwe ukuzinza okulala. Zisetshenziswa ngoba ebusuku-time awakenings, ukuqwasha noma ukuvelela ekuseni.

Uvala ukusetshenziswa

Njengayo yonke imithi, izidakamizwa "Zolpidem" imfundo okuyinto kuqukethwe iphakethe of amakhadibhodi, has Izimo yayo. Umuthi akukashicilelwa ngoba:

  • yokungezwani komzimba ukuze zolpidem noma kwamanye benzodiazepines;
  • nokuvaleka kwemigudu yokuphefumula noma okunzima imvelo acute;
  • ukulala zokuphelelwa umoya ;
  • ukhulelwe;
  • isibindi ezinzima noma izinso;
  • lactation;
  • ukungabekezelelani;
  • abancane.

Kufanele kuphawulwe ukuthi abantu abacindezelekile, kanye notshwala imilutha yezidakamizwa yalabo abaphethwe nezinye izinhlobo ukulutheka, uma uthatha imithi kubhekwe kunesidingo uqaphe kakhulu. Uma kungenjalo, kungenzeka senze isimo sishube nesineke kunzima kangaka.

Yokusetshenziswa

"Zolpidem" ngefomu ithebhulethi ukuze uyiswe nje ngaphambi sokulala. Kusho ukuthi umthamo iyunithi - 10 mg ngosuku. Ukuze umthamo abadala kokuqala kungaba 5 mg. Lapho ngampela ke kungenziwa kabili.

Sangemihla ubuningi "Zolpidem" 10 mg. Isikhathi isicelo kumele singeqi inyanga eyodwa.

Abantu ne lezivakashi ukuqwasha odokotela batusa ukusetshenziswa kwezidakamizwa izinsuku 2-5, futhi isimo - amahora 14-21.

Esimweni lapho ukwelashwa "Zolpidem" luthatha izinsuku eziningana, imithi kungenziwa yema. Uma indlela yokuyelapha ngesonto ezingaphezu kweyodwa, bese ukunciphisa umthamo kufanele kube kancane kancane, ukuze ugweme ukuthuthukiswa ukusabela ezingezinhle.

ohlangothini-imithelela uhlamvu

Njengoba ibekezelelwe izidakamizwa "Zolpidem"? Yokusetshenziswa, ukubuyekezwa bathi ezimweni eziningi angabhekwa umuthi akakubangeli ukusabela ezingezinhle. Nokho, kunezimo lapho ngemuva ukusetshenziswa kwalesi izidakamizwa isiguli namanje azizwa miphumela elandelayo engathandeki:

  • isicanucanu, ukozela, ukuhlanza, ikhanda elibuhlungu, uhudo,
  • ukuqwasha nakuba umuzwa ubuhlungu esiswini, le excitation;
  • isiyezi, amaphupho amabi, ukulahlekelwa amandla okukhumbula kuyinto anterograde (ingozi wale mithandazo ngqo wakhona umthamo akuvumelekile).

Kufanele wazi futhi ukuthi kakhulu kuyaqabukela "Zolpidem" le nkinga ibangelwa elandelayo:

  • ukucasuka, ukudideka, dysphoria, ubudlova;
  • ukusabela engavamile zokuziphatha, somnambulism, sezidakamizwa;
  • ukuqubuka kwesikhumba, izinkinga isibindi emsebenzini, ukuqubuka, ama-enzyme isibindi iyokhushulwa, angioedema;
  • ukuba buthakathaka kwezicubu, itchiness, kwehle izenzo zobulili, urticaria;
  • ataxia, diplopia.

amacala ukweqisa izidakamizwa

Yiziphi izimpawu ukweqisa izidakamizwa kungabangela izidakamizwa "Zolpidem"? Imiyalelo isicelo ibika ukuthi ukuhlukunyezwa olucutshungulwayo imithi noma ngephutha kugwinywe sebuningini amaphilisi isiguli bangezwa ukudideka, ataxia, nobunzima bokuphefumula, ephansi blood pressure, ikhoma nokudideka.

Ngo nesineke ukweqisa izidakamizwa kufanele ngokushesha ngangokunokwenzeka ukuba ahlanze (kungakapheli amahora). Futhi ethintekile kuyadingeka ukunikeza chelators.

Kuleso simo, uma isiguli aquleke, wageza esiswini esebenzisa uphenyo, kanye ukukhiqiza therapy okunezimpawu.

Ukuxhumana nezinye izidakamizwa

Ingabe kuyamukeleka ukuthatha namanye imithi izidakamizwa "Zolpidem"? Yokusetshenziswa (isithako somuthi nokusetshenziswa kwawo ukuthenga lokhu imithi kumele babhale kuphela udokotela abanolwazi) uthi ithuluzi ezifana "Ketoconazole" uyakwazi okuyinani eliphindwe cishe kabili ukwanda nenxenye ukuphila zomuthi. Ngaphezu kwalokho, i-nomuthi kungaba ngcono umphumela CNS ukucindezeleka.

Okhunye okukhambisana imithi ngotshwala ngokuvamile kuholela umphumela okulalisayo zomuthi, kanye ukweqisa izidakamizwa zakhe.

Medicine "rifampicin" kakhulu ngesivinini umzimba, kunciphisa ukusebenza kanye lokuhlushwa amaphilisi.

isabelo ngokucophelela

Yini imithi kufanele imithi ngokuqapha "Zolpidem" okunqunyiwe? Yokusetshenziswa (kusho analogs ezibalwe ngezansi) ibika ukuthi umphumela lokwelapha lungaba ngcono khona omubi, uma izidakamizwa kubhekwe kuhlanganiswe:

  • anxiolytics, barbiturates, izidakamizwa antiepileptic futhi analgesics kwelashwa;
  • izidakamizwa okuyiluthayo, antipsychotics, liphakathi wenza izidakamizwa antitussive kanye nemithi yokunciphisa ukucindezeleka;
  • antihistamine ukuze sedating, izidakamizwa ngoba ukubulawa kwezinzwa okuvamile;
  • "Pizotifenom", "baclofen" futhi "thalidomide".

Kufanele futhi wazi ukuthi ngokuhlanganisa le izidakamizwa nge "buprenorphine" Ngokuphawulekayo kwandisa ingozi yokucindezeleka sezikhungo zokuphefumula.

Izidakamizwa "Zolpidem" nge "itraconazole" bavunyelwe ukuba sihlanganise, kodwa ngokucophelela okukhulu, njengoba kulokhu, ungakwazi ukushintsha izindawo pharmacodynamic futhi pharmacokinetic izindlela kuqala.

ulwazi oluthile

Yini odinga ukuyazi mayelana izidakamizwa "Zolpidem"? Yokusetshenziswa (ezibhebheni lesi sakhiwo okuthengiswa cishe yonke drugstores) uveza ukuthi ukwelashwa eside (cishe 20-30 izinsuku), isiguli singase ukuthuthukisa kwencika ngokwengqondo noma ngokomzimba emuthini. ukusabela okufanayo ichayeke ngokukhethekile labo uke waphawula ukuthi uncike utshwala kanye nezinye izinto. Kule ndaba, iqembu iziguli kufanele igcinwe kokubuyekezwa njalo, futhi ngezikhathi ezithile elibukhali isimo sabo ngokwengqondo nangokomzimba.

Kufanele kuqashelwe ukuthi ingozi sokuncika kwandisa kakhulu uma sicabangela izindlela zihlangana kanjani nezinye benzodiazepines.

Lapho ethola "Zolpidem" nesineke kumele kubhekwe ukuthi ngaphakathi 8 amahora emva ukungenisa amaphilisi, kufanele kube ezenza ubuthongo, ngaphandle kwalokho angase ukuthuthukisa anterograde ukulahlekelwa amandla okukhumbula.

Uma ngemva kwamasonto ambalwa yokwelashwa, ukuqwasha kanye ayizange lidlule, isiguli kufanele bakubheke kabusha isimo. Cishe, ukusabela nakuba enjalo is phetho eyinhloko zengqondo.

Esikhathini Inkambo yokwelashwa olucutshungulwayo kushiwo umuntu kumelwe uyeke ekufezeni imisebenzi ezidinga emakamu eliphezulu ukunakwa, kanye nokushayela imoto.

Abanye abantu ku isizinda "Zolpidem" (ikakhulukazi asebekhulile) angagcina engavamile ezibangela ukuziphatha okuyinqaba nezimpendulo engqondo. Kulokhu, kufanele ngokushesha ayeke ukuthatha izidakamizwa.

Ephambi kwezinduna isifo sesibindi izidakamizwa izidakamizwa esebenzayo kungaba buthelela emzimbeni, bese kamuva kuholele imiphumela engathandeki.

Ngokucophelela okukhulu izidakamizwa kufanele libekwe kubantu asebekhulile. Lokhu kungenxa yokuthi babe ingozi eliphezulu ukupholisa futhi miorelaksiruyuschego umphumela engaholela ukuwa futhi ukulimala.

ukuphila eshalofini, ngokuya ukudayiswa, isitoreji

Ngoba izidakamizwa kubhekwa umlutha, ukuba sikuzuze Kufanele ube udokotela. Ukugcina umuthi it is oyifunayo endaweni okuyinto kahle bavikelekile izingane ezingeni lokushisa hhayi ngaphezu kuka-25 degrees. Impilo eshalofini zomuthi sekuyiminyaka emithathu.

izindlela ezifanayo futhi omqondofana

Izidakamizwa ezivame kakhulu ukuqwasha, okuyizinto analogs "Zolpidem" yilezi ezilandelayo: 'Andante', 'Donormil "," Sondoks "," Barboval "," Zopiclone "," Usokhaya "," imovan ".

Ngokuphathelene omqondofana ukuthi ubheke kubo, "Gipnogen", "Ivadal", "Zolsana", "BID", "Snovitel", "Sanval", "Nitrest".

Lactation nokukhulelwa

Ithonya le izidakamizwa kwabesifazane abakhulelwe engakaze wafunda. Nokho, imiphumela izifundo ukuthi sezenziwe emagundaneni laboratory, baphikisa ngokuthi izidakamizwa has a ukusebenza teratogenic. Kule ndaba, imithi "Zolpidem" ngesikhathi sokukhulelwa is hhayi Kunconywa.

Asinakusho ukuthi okuyiluthayo eziningi ezincane ukungena ubisi lwebele. Ngakho-ke lactation ngesikhathi ukwelashwa kufanele ayeke.

Izibuyekezo Umthengi kanye izindleko izidakamizwa

Thenga izidakamizwa "Zolpidem" kungaba cishe kunoma iyiphi ekhemisi, wemithi nekwetfula somuthi nokusetshenziswa kwawo sikadokotela. Izindleko isilinganiso lomutsi (amaphilisi 10) kuyinto ruble mayelana 820-900. Iziguli bathi kunzima kakhulu inani lentengo eliphezulu okuyiluthayo. Nokho, ochwepheshe libike ukuthi izindleko lokhu umuthi ngempela kulingane, ngoba muhle kakhulu ukuqwasha futhi ubuthongo ompofu. abathengi abaningi ngokuphelele ngokuhambisana nkulumo yokugcina. They phendula kahle imithi, kodwa kufanele iphuzwe ngokuqinile ngaphansi oda udokotela noma imiyalelo.

Kwezokuxhumana yayo, Iziguli asikisela ukuthi izidakamizwa okukhulunywa kubasiza ukuba kahle futhi ngokushesha ukuzumeka futhi ulale kahle ngemuva kokuxinwa ukucindezeleka. Nokho, "Zolpidem" Tablets babe nemiphumela ethile engathandeki. Ngokwesibonelo, bangase baxabane enqabayo okuvame ukuthuthukisa ngesikhathi hypersensitivity kuya asebenzayo izidakamizwa into noma azilungile reception imodi. Imiphumela ezivamile enqabayo yilezi: ikhanda, isiyezi, isicanucanu futhi babone izinto ezingekho. Kulokhu, isiguli singase nomkhuba, ikakhulukazi uma kuhlangene utshwala izidakamizwa.

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