ImpiloAmalungiselelo

"Unitiol": yokusetshenziswa, ngempela

Heavy ubuthi metal, utshwala abampofu kanye nezinye izinto okufanele aphathwe ngokushesha. Uma kungenjalo, kungaholela ekufeni.

izinkampani yesilungu yanamuhla ukwenza okuningi ngokukhishwa kobuthi egazini izindlela. Ziyakwazi kudingekile sokuhoxiswa okusheshayo compounds amagesi anobuthi avela emzimbeni womuntu, kakhulu lula isimo sayo.

Ikhambi ezidume kakhulu ubuthi kuyinto izidakamizwa "Unitiol". Yokusetshenziswa, odokotela impendulo ku ukuphumelela kwalesi imithi kuzoxoxwa ngezansi.

Incazelo, ukubunjwa, uhlobo izidakamizwa ukukhululwa kanye kwikhava yawo,

Ngayiphi ifomu zingatholakala ekhemisi izidakamizwa "Unitiol"? Yokusetshenziswa (ezibhebheni nomuthi is hhayi lwenziwa) ubonisa ukuthi kusho umphenyi ikhiqizwa kunekhambi ecacile okuyinto senzelwe abaphathi ongama noma esicutshini. It has a nephunga eyethile hydrogen sulfide ne ukukhanya color pink (kungenzeka kungenambala).

Yini izingxenye ayingxenye "Unitiol" izidakamizwa? Yokusetshenziswa uthi isithako esebenzayo lokhu ejenti kuyinto dimerkaptopropansulfonat sodium monohydrate. Futhi nomuthi kuhlanganisa kwakwakhe asizayo njengoba sulfuric acid, disodium edetate (Trilon B), namanzi umjovo.

Ngo ukuthengiswa umuthi ihlinzekwa e ingilazi ampoules 5 ml. Agcwele ku nentaba kwengqamuzana, okuyinto ezibekwe inqwaba iphepha.

izakhiwo pharmacodynamic

Kanjani lesi sidakamizwa "Unitiol"? Yokusetshenziswa ibika ukuthi lokhu ejenti ngokukhishwa kobuthi egazini, okuyinto ngempela fast yokugudluza kusilela amaqembu sulfhydryl. Ngokusho mode kwabo isinyathelo lokhu izidakamizwa liseduze kakhulu kompleksonam.

Ngokwe-art, amaqembu sulfhydryl uyakwazi ukusabela nge thiol ubuthi egazini, izicubu, kanjalo zakha isimiso ayinangozi izakhiwo babaleki umchamo.

ubuthi Lock kunomthelela imisebenzi ukubuyiselwa izinhlelo enzyme emangqamuzaneni okuthiwa beshaywa ezinobuthi. Lesi sidakamizwa isetshenziswa kuyindlela yokuvimbela ubuthi by-arsenic, izinsimbi ezisindayo kanye compounds zabo.

Abantu ne polyneuropathy sikashukela kanye nesisekelo-amyloidosis yesibili le nomuthi kunciphisa ubuhlungu, ngcono ukusebenza weSigungu Sikazwelonke, futhi ulawula permeability ka-capillary.

izici kinetic

Yiziphi izindawo esingokwemvelo kinetic we nomuthi "Unitiol"? Yokusetshenziswa ugomela ngokuthi emva umjovo ongama noma esicutshini engqamuzaneni izidakamizwa ngenkuthalo lingene egazini. Ubuningi esiphezulu izidakamizwa kulotshwe ngemva cishe 40 imizuzu (emva / m).

Isigamu-ukuphila amathuluzi kuyinto amahora amabili. Kuncike izidakamizwa umchamo ngesimo imikhiqizo ngokwengxenye namachibi.

isixazululo izinkomba

Ngaphansi Inikeza buphi ubufakazi bokuthi isiguli angabelwa ukuba umuthi "Unitiol"? Yokusetshenziswa (imijovo kufanele sigcwaliswe kuphela lochwepheshe bezokwelapha abanolwazi) ubonisa ukuthi leli thuluzi isetshenziselwa:

  • ukudakwa bismuth arsenic, i-chromium, mercury noma glycosides inhliziyo;
  • utshwala, kanye nemvelo ezingamahlalakhona of delirium oludakayo njengengxenye ukwelashwa;
  • ukonakala gepatotserebralnoy (Wilson syndrome).

Izimo izidakamizwa

Ingabe kukhona Izimo kule izidakamizwa "Unitiol"? Iziyalezo yokusetshenziswa ithi ayikwazi kubhekwa indlela yokunika ku:

  • sensitization emuthini;
  • yokwehluleka kwesibindi ukusebenza;
  • njengoba ingane;
  • ukhulelwe;
  • nomfutho wegazi ophezulu;
  • ibele.

Izidakamizwa "Unitiol": yokusetshenziswa

I ampoule iyithuluzi angathengwa ngasiphi ekhemisi. Ngokusho imiyalelo, umuthi kumele phansi kwesikhumba iqondiswa noma intramuscularly.

Ekwelapheni arsenic ukudakwa nomuthi isetshenziswa ngesilinganiso 50 mg isithako esebenzayo ngayinye 10 kg isisindo umzimba isisulu (isb 250-500 mg). Ngosuku lokuqala ukwelashwa wabonisa Isikali kufanele sinikezwe kuze kube izikhathi 4, okwesibili - izikhathi 3, kanti elandelayo - kanye.

Ekwelapheni mercury poisoning nosawoti nomuthi isetshenziselwa isikimu ngenhla echazwe izinsuku eziyisikhombisa noma kwaze kwaba yilapho zinyamalala ephelele izimpawu zokudakwa.

Ekwelapheni ushevu glycosides inhliziyo ngosuku lokuqala nelesibili kwezidakamizwa iqondiswa ngesilinganiso 50 mg isithako esisebenzayo ngayinye 10 kg isisindo isiguli (ngamanye amazwi, 250-500 mg) kane ngosuku, futhi ngosuku olulandelayo - kabili noma kuze izimpawu cardiotoxicity.

Therapy gepatotserebralnoy sokuwohloka nomuthi iqondiswa intramuscularly at 5.10 ml lokuhlushwa ejwayelekile nsuku zonke noma masonto kwezinsuku ezimbili. Isikhathi yokuyelapha 26-30 imijovo. Uma kudingeka, ukuphinda Yiqiniso ngemuva kwezinyanga 4.

Ukuze ekwelapheni ezingamahlalakhona ukulungiselela ukusebenzisa uphuzo ngokweqile uhlamvu lisetshenziswa inani 4-5 ml lokuhlala ejwayelekile kuze kube izikhathi 3 ngesonto.

Ekwelapheni delirium, le nomuthi iqondiswa kanye (5 ml lokuhlushwa ejwayelekile)

side effects

Ngo nesicelo esicutshungulwayo enqabayo izidakamizwa ukusabela zenzeka kakhulu akuvamile. Kwezinye izimo, isiguli athuthukile tachycardia, isiyezi, isicanucanu futhi isikhumba pallor. Ngaphezu okungenhla, bangase baxabane nomzimba.

Overdose nezidakamizwa ekuxhumaneni

Endabeni ka ukweqisa izidakamizwa, isiguli iphika, hyperkinesis, retardation, ukuquleka, futhi ukucobeka. Kulokhu, ukwelashwa lingaze.

Lesi sidakamizwa aluhambisani ne-ejenti pharmacologically zihlanganisa izinsimbi ezisindayo, kanye lezisekelo. Futhi ke akuyona enikezwa "Acizol".

Izibuyekezo

Umthengi Izibuyekezo yokucabangela kusho ivelakancane. Lokhu kuhlobene kakhulu iqiniso lokuthi le nomuthi is mhlawumbe kusetshenziswa umkhuba umile.

Njengoba odokotela abanolwazi, bakhuluma "Unitiol" isixazululo njengoba esebenza kahle kakhulu futhi ngempumelelo izindlela okuyinto evacuates ubuthi, kuhlanganise e ubuthi oludakayo.

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