ImpiloAmalungiselelo

Naiz (tablet) - imfundo manual.

ifomu Isikali

Ukulungiswa senziwa amafomu 3-izidakamizwa - ukumiswa, amaphilisi dispersible futhi ezivamile. Ukumiswa kunuka kamnandi mfana zokunambitha ephuzi ngombala futhi ngempela nobuntu lokhu izidakamizwa. Ukumiswa kungenziwa redispersed by shaking isitsha.

Tablets ekhiqizwa awube mhlophe, ephethe tinge kancane aphuzi. Izibhebhe ukuma isiyingi, biconcave, evele yayo kokubili iyashelela.

Nise Ukwakheka:

ukumiswa

izidakamizwa okusebenzayo

  • Nimesulide - 50 mg (5 ml ukumiswa)

Excipients:

  • sorbitol
  • glucose
  • gum xanthan
  • propyl
  • methylparaben
  • citric acid
  • uphayinaphu flavour
  • Yellow udayi WS
  • glycerol
  • polysorbate
  • manzi ahlanzekile

amaphilisi dispersible

izidakamizwa okusebenzayo

  • Nimesulide - 50 mg (Table 1).

excipients

  • aspartame
  • calcium phosphate
  • microcrystalline cellulose
  • carboxymethyl isitashi
  • corn isitashi
  • talc
  • magnesium stearate
  • Colloidal Silicon dioxide
  • uphayinaphu flavour

amaphilisi

izidakamizwa okusebenzayo

  • Nimesulide - 100 mg (Table 1).

Excipients:

  • magnesium stearate
  • Calcium Hydrogen Phosphate
  • microcrystalline cellulose
  • Anhydrous Silicon colloidal
  • corn isitashi
  • Sodium isitashi glycolate
  • talc ukuhlanzwa

Isenzo kwemithi zomuthi

isinyathelo kwemithi uyalandisa ngokuyinhloko Nise - amaphilisi ami, ukulaya iphethe imininingwane zonke izinhlobo umthamo. Umuthi kuyinto NSAID, eliqukethe e isakhiwo sulfonilidnuyu yayo ngamaqoqo. may Nimesulide iphathelene inhibitor of Cox-2, ukuze kunemiphumela eqeda ukuvuvukala kanye analgesic, ngaphezu, umuthi uzabalaza nemiphumela analgesic, kodwa kancane.

Lo mshini wezenzo zomuthi elihlobene ne nokucindezela synthesis prostaglandins e ukuvuvukala nokucindezela kumiswa-mpilo ezizivelelayo kanye okusithiyayo of myeloperoxidase ukukhululwa.

Pharmacokinetics

Nise ugxile ngokuphelele kusukela ipheshana emathunjini, ukufinyelela esiphezulu yayo egazini kakade emva kwamahora angu-2. Umuthi kuyinto 99% amaprotheni eboshiwe.

Ukulungiselela nize - amaphilisi Umhlahlandlela esithathelwe imithombo ezisemthethweni, metabiliziruetsya esibindini futhi excreted ku umchamo, u-98% umthamo eyamukelwe okukhipha emini.

ubufakazi

  • izifo Rheumatic ukuthi ukuthuthukisa ngaphandle egobolondweni lelunga
  • osteoarthritis
  • Ukuvuvukala nobuhlungu emva kokuhlinzwa
  • Nobuhlungu obubangelwa dysmenorrhea
  • Imfiva ubuhlungu ngesikhathi ukuvuvukala acute e yomoya engenhla

Imiphumela engemihle Nise

Tablets, isiqondiso lapho manje, ungaveza ohlangothini-imiphumela kumasistimu ahlukahlukene kanye nezinhlaka:

imiphumela emibi izidakamizwa, ezihlobene ipheshana yesisu

  • isicanucanu
  • isilungulela
  • ubuhlungu esiswini
  • hlalani indle

imiphumela emibi izidakamizwa, ezihlobene isimiso sezinzwa esiyinhloko:

  • ubuhlungu bekhanda
  • ukozela
  • isiyezi

imiphumela emibi izidakamizwa, ezihlobene komzimba:

  • erythema
  • ukuqubuka
  • urticaria

Eminye imiphumela emibi:

  • Ukugcinwa oketshezini lomzimba
  • oliguria
  • ukuvuvukala

Izimo Nise

Ingabe uhlu Izimo lapho kunconywa ukugwema ngokuthatha izidakamizwa, futhi uma kudingekile, kuphela emva kokubonisana udokotela wakho.

  • Ukopha kusukela ipheshana emathunjini
  • ukungasebenzi kwezinso
  • ukuhluleka hepatic
  • Nokukhulelwa kanye lactation
  • Peptic nezifo zesisu

Izidakamizwa nokuxhumana nize

Tablets, imiyalelo ukusetshenziswa okungadingi kuholele idatha ephelele neqondakalayo ku konke ukuhlanganyela izidakamizwa ekwakhiweni lalithé: hhayi Kunconywa ne ejenti ezilandelayo - phenytoin, digoxin, iyiphi isisu, izidakamizwa lithium, anticoagulants, izidakamizwa antihypertensive, ama-NSAID, methotrexate, cyclosporin .

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