Impilo, Amalungiselelo
Naiz (tablet) - imfundo manual.
ifomu Isikali
Ukulungiswa senziwa amafomu 3-izidakamizwa - ukumiswa, amaphilisi dispersible futhi ezivamile. Ukumiswa kunuka kamnandi mfana zokunambitha ephuzi ngombala futhi ngempela nobuntu lokhu izidakamizwa. Ukumiswa kungenziwa redispersed by shaking isitsha.
Tablets ekhiqizwa awube mhlophe, ephethe tinge kancane aphuzi. Izibhebhe ukuma isiyingi, biconcave, evele yayo kokubili iyashelela.
Nise Ukwakheka:
ukumiswa
izidakamizwa okusebenzayo
- Nimesulide - 50 mg (5 ml ukumiswa)
Excipients:
- sorbitol
- glucose
- gum xanthan
- propyl
- methylparaben
- citric acid
- uphayinaphu flavour
- Yellow udayi WS
- glycerol
- polysorbate
- manzi ahlanzekile
amaphilisi dispersible
izidakamizwa okusebenzayo
- Nimesulide - 50 mg (Table 1).
excipients
- aspartame
- calcium phosphate
- microcrystalline cellulose
- carboxymethyl isitashi
- corn isitashi
- talc
- magnesium stearate
- Colloidal Silicon dioxide
- uphayinaphu flavour
amaphilisi
izidakamizwa okusebenzayo
- Nimesulide - 100 mg (Table 1).
Excipients:
- magnesium stearate
- Calcium Hydrogen Phosphate
- microcrystalline cellulose
- Anhydrous Silicon colloidal
- corn isitashi
- Sodium isitashi glycolate
- talc ukuhlanzwa
Isenzo kwemithi zomuthi
isinyathelo kwemithi uyalandisa ngokuyinhloko Nise - amaphilisi ami, ukulaya iphethe imininingwane zonke izinhlobo umthamo. Umuthi kuyinto NSAID, eliqukethe e isakhiwo sulfonilidnuyu yayo ngamaqoqo. may Nimesulide iphathelene inhibitor of Cox-2, ukuze kunemiphumela eqeda ukuvuvukala kanye analgesic, ngaphezu, umuthi uzabalaza nemiphumela analgesic, kodwa kancane.
Lo mshini wezenzo zomuthi elihlobene ne nokucindezela synthesis prostaglandins e ukuvuvukala nokucindezela kumiswa-mpilo ezizivelelayo kanye okusithiyayo of myeloperoxidase ukukhululwa.
Pharmacokinetics
Nise ugxile ngokuphelele kusukela ipheshana emathunjini, ukufinyelela esiphezulu yayo egazini kakade emva kwamahora angu-2. Umuthi kuyinto 99% amaprotheni eboshiwe.
Ukulungiselela nize - amaphilisi Umhlahlandlela esithathelwe imithombo ezisemthethweni, metabiliziruetsya esibindini futhi excreted ku umchamo, u-98% umthamo eyamukelwe okukhipha emini.
ubufakazi
- izifo Rheumatic ukuthi ukuthuthukisa ngaphandle egobolondweni lelunga
- osteoarthritis
- Ukuvuvukala nobuhlungu emva kokuhlinzwa
- Nobuhlungu obubangelwa dysmenorrhea
- Imfiva ubuhlungu ngesikhathi ukuvuvukala acute e yomoya engenhla
Imiphumela engemihle Nise
Tablets, isiqondiso lapho manje, ungaveza ohlangothini-imiphumela kumasistimu ahlukahlukene kanye nezinhlaka:
imiphumela emibi izidakamizwa, ezihlobene ipheshana yesisu
- isicanucanu
- isilungulela
- ubuhlungu esiswini
- hlalani indle
imiphumela emibi izidakamizwa, ezihlobene isimiso sezinzwa esiyinhloko:
- ubuhlungu bekhanda
- ukozela
- isiyezi
imiphumela emibi izidakamizwa, ezihlobene komzimba:
- erythema
- ukuqubuka
- urticaria
Eminye imiphumela emibi:
- Ukugcinwa oketshezini lomzimba
- oliguria
- ukuvuvukala
Izimo Nise
Ingabe uhlu Izimo lapho kunconywa ukugwema ngokuthatha izidakamizwa, futhi uma kudingekile, kuphela emva kokubonisana udokotela wakho.
- Ukopha kusukela ipheshana emathunjini
- ukungasebenzi kwezinso
- ukuhluleka hepatic
- Nokukhulelwa kanye lactation
- Peptic nezifo zesisu
Izidakamizwa nokuxhumana nize
Tablets, imiyalelo ukusetshenziswa okungadingi kuholele idatha ephelele neqondakalayo ku konke ukuhlanganyela izidakamizwa ekwakhiweni lalithé: hhayi Kunconywa ne ejenti ezilandelayo - phenytoin, digoxin, iyiphi isisu, izidakamizwa lithium, anticoagulants, izidakamizwa antihypertensive, ama-NSAID, methotrexate, cyclosporin .
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