Impilo, Amalungiselelo
"Fokusin": ukubuyekezwa odokotela, contraindications yokusetshenziswa
Uyini izidakamizwa "Fokusin"? Uphenyo odokotela, contra-izinkomba, futhi lokhu kusho ukuthi ngeke ukwethula izinto kwalesi sihloko. Kusukela ke uzofunda ngalokho lokhu izidakamizwa anezakhi, ifomu lapho kukhiqizwa, okubangela yimuphi ukuphendula uhlangothi.
Ubujamo, incazelo, ukwakheka kanye nokupakisha
Yini ifomu owenza izidakamizwa "Fokusin"? Yokusetshenziswa, ukubuyekezwa ukubika ukuthi lokhu izidakamizwa uyadayiswa yini uhlobo kanzima gelatin amaphilisi. Banezinhliziyo umzimba okusobala emnyama cap okwesibhakabhaka.
Zonke amaphilisi Isikali egcwele umbala micropellet omhlophe noma awube mhlophe. nempahla yabo okusebenzayo tamsulosin hydrochloride, kanye nokusekela izakhi copolymer methacrylate ukuhlakazwa isetshenziswa, dibutyl sebacate, microcrystalline cellulose, talc, polysorbate 80 kanye aqueous colloidal Silicon dioxide.
Ngokuphathelene igobolondo capsule, liphethe azorubin, lobunikazi udayi oluhlaza okwesibhakabhaka kanye gelatin.
Thenga le imithi kungaba iziqukathi contoured, okuyinto ezibekwe amabhokisi leyakhiwe ngemabhokisi.
kwemithi
Kuyini izidakamizwa emangalisayo "Fokusin"? Izibuyekezo ukubika ukuthi sihlobana iqembu kwemithi ye-alpha-blocker. Lokhu nomuthi eqondiswa urodynamics futhi sithinta izinqubo umzimba ukuthi kwenzeke wendlala.
Umthelela zokwelapha zomuthi ngenxa izithako ezisebenzayo e ngezithako zawo.
Njengoba kushiwo ngenhla, isithako esebenzayo ye nomuthi izenzo tamsulosin hydrochloride. Le nto powder emhlophe kokuba isakhiwo crystalline. Kuyinto kahle oncibilikayo emanzini, kancane oncibilikayo ethanol futhi glacial acetic acid, futhi cishe zingaxazululeki ether.
Izici imithi
Yiziphi izinto ezinganembile esivela izidakamizwa "Fokusin"? Yokusetshenziswa, ukubuyekezwa ukubika ukuthi leli thuluzi uyakwazi ukuvikela i-alpha-receptor, okuyinto yenziwe yaba yasendaweni ku ulwelwesi postsynaptic. Futhi, lokhu kuvimbela ukudlula nomuthi ngokusebenzisa pulses vasoconstrictive synapse adrenergic, okubangela ukunwetshwa precapillaries futhi arteriole.
Omunye umphumela umuthi tamsulosin hydrochloride ikhono ukuvimba-alpha-receptor 1-adrenergic zitholakala ezindaweni Prostatic, futhi enemisipha esinyeni igobolondo. ukuchayeka esinjalo sithuthukisa imingcele urodynamic, ikakhulukazi umdlavuza wendlala.
izakhiwo
Ngemva kwesikhathi esithile kuboniswe ukusebenza emitholampilo "Fokusin" izidakamizwa? Uphenyo odokotela bathi umphumela lokhu izidakamizwa ephawuleka izinsuku ezingu-14 kuphela ngemva Ukuqalwa yokwelapha.
Nakuba ngokuthatha izidakamizwa, iziguli:
- anda urethral inesikhala;
- ukuzinza of kwegazi detrusor;
- ukwandisa mafutha anciphisa isikhala esingaphakathi entanyeni esinyeni;
- ngcono imisipha umzimba esinyeni;
- ekunciphiseni ingcindezi ku urethra;
- wehlise zamanje umchamo ukumelana;
- ukuzinza of ukuchama;
- ehle kobukhulu izimpawu yokucasuka, okuyinto zibangelwa adenoma we wendlala;
- wehlise esengezweni izimpawu isimiso urinary.
Kufanele kuqashelwe ukuthi le izidakamizwa okukhulunywa akakubangeli ukunciphisa umfutho wabo wegazi.
Pharmacokinetics
Uyini kinetic imingcele imithi "Fokusin"? Izibuyekezo odokotela (Izimo izidakamizwa izokwethulwa ngezansi) sibeke ukuthi inqubo ukuncela wenziwa tamsulosin hydrochloride e pheshana emathunjini. Umsebenzi esiphezulu ebonwe ukumuncwa lapho izidakamizwa sathathwa ngemva kokudla.
I bioavailability efana 100%. Ngemva umthamo owodwa we izidakamizwa, esiphezulu yayo waphawula plasma lokuhlushwa amahora 6.
isimo Esimile kufinyelelwa nesineke emva kwezinsuku 5 nokushintsha kokudla nokufakwa okuqhubekayo.
izidakamizwa umzimba uyephuza kakhulu. It is excreted ku umchamo
ubufakazi
Yini izidingo eyethulwe izidakamizwa? Kuthiwani lo mbiko ubukeza wezokwelapha? "Fokusin" Tablets dizuricheskih engabelwe ekwelapheni iziyaluyalu okuyinto zibangelwa adenoma we wendlala.
Lo muthi kufanele athathwe kuphela ngemva kokukhuluma nodokotela.
Izimo
Kungaphansi kwaziphi izimo akusho linqume izidakamizwa ukuze Fokusin iziguli ' "? Uphenyo odokotela (Izimo kwaleli thuluzi izokwethulwa Manje) umbiko ukuthi ukuvinjelwa kuxoxa ngazo cishe akukho imithi. It ayikwazi ukusetshenziswa uma hypersensitivity kuya izingxenye asebenzayo nasizayo, kanye hypotension orthostatic.
Ngokucophelela okukhulu, lokhu izidakamizwa ezinqunyiwe ukuze abantu ukwehluleka ezinzima kwezinso futhi hepatic.
Izidakamizwa "Fokusin": isitatimende
Izibuyekezo Ochwepheshe ukubika ukuthi umthamo kahle le izidakamizwa abadala 1 capsule ngosuku.
Umuthi Kunconywa ukuthatha ngokushesha ngemva kokungenisa kuqala. I capsule kufanele kugwinywe lonke hhayi baba imilutha ye.
side effects
Zikhona yini imiphumela emibi kwenzeka seziguli ezithola "Fokusin" izidakamizwa? Iziguli amazwana ngokuvamile aqukethe izikhalazo mayelana ezifana izenzakalo engathandeki njengoba:
- isiyezi, nokulahlekelwa ukwazi, ikhanda;
- hypotension postural, tachycardia;
- ukungasebenzi umgudu wokuphefumula (rhinitis);
- ukukhungatheka ngezinsimbi zesihlalo, ukuhlanza, isicanucanu;
- ukushayisana kohlelo zokuzala.
Bangase abonise ezifana side effects njengoba sokukhathala esingamahlalakhona futhi pupillary constriction.
amacala ukweqisa izidakamizwa
Uma weqa umthamo watusa zomuthi "Fokusin" kunobungozi enkulu yokuba izimpawu ka-acute lwemithambo hypotension. Kulokhu, isiguli kufanele afune usizo lodokotela.
Ukwelapha isimo esiswini wahlupheka sagezwa namalahle isebenze.
izidakamizwa ekuhlanganyeleni
Nge inhlanganisela "Fokusina" nezidakamizwa antihypertensive ne-beta-blocker akukho ukuxhumana lezi zimali akufanele kumakwe.
ekuphathweni esisodwa zomuthi nge antiulcer izidakamizwa kubangela ukwenyuka emakamu plasma wokuqala. Umthelela ukubuyela emuva zile uma ukudlala "Fokusina" nge isisu.
Ngokwe-art, umuthi okukhulunywa uyakwazi ukusabela nge:
- ejenti hypoglycemic;
- tricyclic antidepressant;
- bronchodilators izidakamizwa;
- izidakamizwa hormone anticancer.
Inani kanye analogue
Have izakhiwo efanayo izidakamizwa ezifana "Tamsol", "Adenorm", "Flosin", "Bazetu", "Urofrin", "Omiks", "Tulozin" "Omnic", "Taniz", "Omnimaks" "Tamsulosin "" Ranoprost "," Tamsonik "," Tameks ".
Izindleko isilinganiso "Fokusin" izidakamizwa kuleli zwe uyahluka ruble 480-500 ngoba amaphilisi 30 futhi ruble 1000-1200 ngoba amaphilisi 90.
Uphenyo nomuthi
Iningi leziguli ezine-umdlavuza wendlala noma wendlala bephoqeleka ukuba ngidle izidakamizwa namalungu tamsulosin. Ukuhlaziya izimpendulo zabo, singaphetha kahle ngokuthi iningi lawo uthanda izidakamizwa kuka nozakwabo zayo.
Ukukhetha phakathi izindlela ezifana "Omnic" noma "Fokusin" amadoda amaningi makudle kwabo ukhetho lwesibili. Zithi kungenzeka avuse onjalo engemihle effect okuningi kancane ejaculation retrograde.
Phakathi ukubuyekezwa omuhle odokotela yiwo evame kakhulu, othi ukuqokwa kweziguli amaphilisi ka ukuchama eyeka ekuletheni izinkinga. Ngaphezu kwalokho, wokuphuthuma ukuba kunyamalale ngokuphelele.
Manje uyazi ukuthi kuyinto izidakamizwa "Fokusin". Uphenyo odokotela, contra-izinkomba kanye izidakamizwa ezichazwe kulesi sihloko. Kumele wakhumbula ukuthi linqume lokhu izidakamizwa kufanele kuphela kube abanolwazi lochwepheshe.
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