Impilo, Amalungiselelo
Umuthi 'Somnol ": yokusetshenziswa, analogs, ukubuyekezwa
Abaningi bethu okungenani kanye empilweni yakhe yayinezinkinga yobuthongo. Uma kwaba ngawe kuyinsakavukela futhi kuphazamisa zokuphila kwansuku zonke, singasho ngokuphepha ukuthi ukucasula yemvelo inqubo bokuphila, uhlale usesimweni nge eliphansi umsebenzi ubuchopho futhi impendulo ethambile ukuze kwezwe elisizungezile. Ngenxa ukulala thuthuva avele hhayi kuphela ukozela, kodwa futhi eziwohlokayo ibhalansi engqondo kanye nezempilo. Uma uneminye izinkinga zalolu hlobo, ufika izidakamizwa ethi "Somnol". Izinkomba ukusetshenziswa, incazelo isenzo kwemithi, odokotela yangempela kanye neziguli, kanye kungekho analogue izidakamizwa kancane ngempumelelo Kuxoxwa le nto.
ifomu Isikali kanye nokusungulwa
A ukulungiselela inethiwekhi ekhemisi kuyinto ngesimo amaphilisi biconvex ezimhlophe camera ohlangothini phambi okuyinto kukhona ingozi. Basuke zahlanganiswa ngo amabhamuza yizicucu 10. Kokunye ithebhulethi "Somnola" iqukethe 7.5mg ka zopiclone, amazambane isitashi, magnesium stearate, anhydrous calcium hydrogenphosphate, sodium glikopat, Silica, aerosil, futhi povidone kanye Umbala ejenti.
pharmacodynamics
Ingqikithi eziyisisekelo, ingxenye "Somnola" kuyinto okuyiluthayo, elingelakwaJuda tsiklopirrolonov iqembu. Zopiclone has a okuyiluthayo, sine anticonvulsant, tranquilizing futhi imisipha relaxant imiphumela. Le miphumela kwemithi ngenxa isenzo efana zokungabi receptor we isimiso sezinzwa esiyinhloko.
Lapho ethola izidakamizwa, izidakamizwa eyisisekelo zopiclone encishisiwe isikhathi sokulala futhi imvamisa awakenings nasebusuku, kukhuphuke ubuthongo ubude kanye izinga.
Ukuze ukwelashwa isikhathi eside, kuze kufinyelele ezinyangeni 4 ngaphandle izidakamizwa eziluthayo "Somnol" (incwadi yeziyalezo ibonisa ukuthi leli).
imiphumela kwemithi
Umehluko omkhulu phakathi 'Somnola "kusuka kwamanye amaphilisi elele - khona ukubunjwa yayo ekhuthaza zamakhemikhali ezibizwa ngokuthi zopiclone. Lokhu kusho ukunciphisa isikhathi ukuzumeka, uma isekela ubuthongo kuqala, ngaphandle kokuphazamisa shift isigaba futhi izinga layo. Umthelela izidakamizwa kwenzeka ngaphakathi isigamu sehora ngemuva kokwemukelwa yayo futhi kuthathe amahora 6-8, okuyinto ezokwenzeka ubude evamile, yemvelo inqubo bokuphila, uhlale esitha, isimo sakugcina umsebenzi ubuchopho futhi impendulo sehliselwe kwenzekani emhlabeni.
Cishe ingekho lapho ithola "Somnol" izidakamizwa ngokungafani barbiturates futhi benzodiazepines, ukozela nobuthakathaka. Yokusetshenziswa ibonisa ukuthi isigamu-ukuphila umzimba ingeqi amahora 3.5-6, ngisho ukusetshenziswa isikhathi eside, metabolites kungukuthi cumulated. Izibuyekezo abonisa ukuthi leli thuluzi aqede ubuhlungu bekhanda kubantu somoya lapho ithola imvamisa ukuncipha ebusuku futhi ekuqaleni kuka ukuhlaselwa ekuseni, kanye ubude babo kanye ngamandla.
Izidakamizwa "Somnol": imfundo, izinkomba ukusetshenziswa
Kwezinye izimo, ukuze kuxazululwe izinkinga ukusetshenziswa imithi? Izidakamizwa "Somnol" manual uncoma ukusetshenziswa uma:
- izinkinga zokulala eyisisekelo (nobunzima ngilale, awakenings njalo ebusuku, futhi isimo lezivakashi ukuqwasha ifomu).
- isifuba somoya bronchial, esibonakala by neziqubu ebusuku ekuseni. Ithathwe ngokuhlanganyela "theophylline".
- iziyaluyalu yesibili zilale zengqondo.
Umthamo nokuPhatha
Udle isidakamizwa "Somnol" (manual kubonisa lokhu). Sebenzisa imithi Kunconywa emfushane, kwamasonto 4, kucatshangelwa inkathi umthamo ukunciphisa. Khulisa isikhathi yokwelapha kungenzeka kuphela ngemuva kabusha nokuhlola nesineke.
Ukwelashwa kufanele uqale nge umthamo ubuncane, noma kunjalo akufanele sedlule ngemithamo kuvunyelwe.
Izidakamizwa "Somnol" imfundo manual incoma ukuthatha ikakhulukazi ngesikhathi sokulala.
Endabeni ekwelapheni izifo izinso ukuqala amaphilisi isigamu (3.75 mg), naphezu kweqiniso lokuthi ekuqongeleleni zopiclone futhi metabolites ningagcini ukuhluleka kwezinso.
Iziguli kuze iminyaka 65, lesi sidakamizwa "Somnol" afundiswe izibhebhe 7.5 mg Kunconywa ukuthatha kanye ngosuku.
Uma kwephulwa kwesibindi, impatho isiqalisile nge 3,75 mg hhayi ngaphezu kwesikhathi esisodwa ngosuku, ngoba isikhathi kwezidakamizwa excretion ezigulini enjalo kuyehla. Uma kudingeka, umthamo kungase kukhule ku-7.5 mg, kuyilapho ngempela kucatshangelwe ukuzwela umuntu ukuba izithako izidakamizwa.
Lapho ukwelashwa sekudlulile zokucindezeleka zokuphefumula, kanye kahle isibindi umsebenzi, uqala nge 3,75 mg hhayi ngaphezu kwesikhathi esisodwa ngosuku. Le nqubo ibizwa futhi esetshenziselwa abantu abaneminyaka engama-65, umthamo kungenziwa kancane kancane uma kudingeka.
Kungakhathaliseki izimpawu I-"Somnol" izidakamizwa, umthamo wansuku zonke akufanele bube ngaphezu kuka-7.5 mg. Lapho izivakashi ukwelashwa ukuqwasha ihlala izinsuku ezingu-5, futhi uma isimo - kungakapheli amaviki ezingaphezu kwezingu-3. Njengoba for ifomu okungamahlalakhona, esimweni esinjalo onguchwepheshe kuphela kuchazwe Yiqiniso yokwelapha.
izidakamizwa ekuhlanganyeleni
Nakuba yokuvuma "Somnol" imithi nge neuroleptics, ezinye izindlela okuyiluthayo, anticonvulsant futhi sine-zinhlungu, imithi yokucindezeleka nezidambisa analgesics opioid, imithi ebulala izinzwa, noma erythromycin sithuthukiswe nokudangala nomthelela isimiso sezinzwa esiyinhloko.
Ekwelapheni ngokuvumelana nomuthi e emakamu plasma kunciphisa trimipramine futhi buthakathaka umphumela wawo.
Izidakamizwa "Somnol" imfundo manual sivimbela ukusetshenziswa ngokuhlanganyela Ethanol ngoba kungabangela ukupholisa inzuzo phansi izidakamizwa - zopiclone.
side effects
Ochwepheshe bezifo, kanye nokwelashwa nesineke "Somnolom" kungase kuhambisane miphumela elandelayo engathandeki:
- Kwemizwa uhlelo - ukozela, ubuthakathaka ngemva ilele, ikhanda, isiyezi, isimo sokucindezeleka, ukulahlekelwa ikhono ukukhumbula izenzakalo. Ngenxa yalokho isicelo we okuyiluthayo kwezinye izimo avele ukusabela nakuba: ukucasuka, okuyinto angakhula abe nolaka, ukubambisana aphazamiseke ukunyakaza, lokuhlushwa imemori, izinga ukusabela engqondo iba ukwazi bedidekile, ukucindezeleka livela. Uma isiguli uyayeka ngokuthatha izidakamizwa, "Somnol" (imfundo, izinkomba ukusetshenziswa kukhona asendabeni), kungase kube lezivakashi ukuphazamiseka kokulala.
- ipheshana yesisu - esiphazamisayo yokwenza evamile esiswini, kukhona metallic noma ukunambitheka ababayo emlonyeni.
- Laboratory imingcele - e-serum igazi isigqugquzeli transaminases hepatic futhi ane-alikhali phosphatase.
- Amasosha omzimba - kukhona komzimba ezifana urticaria, pruritus, ezimweni ezingajwayelekile - angioedema.
Izimo
Ukusebenzisa izidakamizwa "Somnol" imfundo ayikuvumeli:
- Lapho hypersensitivity kuya izithako.
- Ebusuku stop ukuphefumula ukunyakaza.
- Lokulingene noma okunzima sokuhlasela kwamasosha omzimba nezifo kwamanyuroni.
- Zokuphefumula, esingamahlalakhona kwezinso noma hepatic.
- Ukukhulelwa.
- Ngesikhathi lactation.
Ngaphezu kwalokho, lokhu okuyiluthayo contraindicated ezinganeni ezingaphansi kweminyaka engu-18 ubudala.
Ungakhohlwa ukuthi imithi kungadala ithemba, kukhona futhi ekuthuthukiseni lesi sifo, ngakho akuvumelekile ngaphandle iseluleko wazibonela okwandisa umthamo kanye nesikhathi sokwelashwa.
ukweqisa izidakamizwa
Izimpawu yokudlula umthamo watusa kuxhomeke endleleni umuntu ocindezelekile ngaso isimiso sezinzwa esiyinhloko. Ngokuvamile, somnolence, ngezinye izikhathi umuntu ewela equlekile. Usizo lokuqala kufanele babe nesineke iphume esiswini, thatha namalahle yasebenza, uma kunesidingo, sebenzisa yokwelapha lingaze esibhedlela. Hemodialysis ukweqisa izidakamizwa "Somnolom" ihumusha isenzo ayizwakali. Kuyindlela yokuvimbela ungasebenzisa izidakamizwa kusukela iqembu detoxifying izidakamizwa - "flumazenil".
Izixwayiso
Ukulungiselela "Somnol" (incwadi yeziyalezo, okukala okunemininingwane impahla) kumele bafake iziguli ukunakekelwa okukhethekile nge sezinso futhi izifo zesibindi nasebekhulile. Esikhathini esiyiminyaka ukwelashwa akuvunyelwe nakancane ukuphuza.
Ngaphansi amponjwana ukwandisa umphumela okulalisayo amaphilisi elele. Ukusetshenziswa ahlangene kwala magciwane kubangela ukozela emva uvuka, esithinta ikhono ukushayela imoto.
Reception "Somnola" kungaholela ukuthuthukiswa sokuncika ngemilingo nokungokwenyama. Ezimweni ezinjalo ezingavamile kakhulu, lapho kwelashwa esingangenyanga. Uma umthamo kanye nesikhathi nokuphathwa izidakamizwa abangu ngokuzimela anda ematfuba kwencika iyakhula.
Sizonyuka ingozi nge izimali zosizo aphoyintimenti abantu abanale nkinga yokungadli kahle ubuntu kanye umlando we utshwala ngokweqile kanye nokulutheka ngemithi ethile. ukuqedwa ngokuzumayo okuyiluthayo in iziguli ukuluthwa kungabangela ekuthuthukiseni lesi sifo, okuyinto libhekene ukuvela imizwa yokwesaba, ikhanda kanye ubuhlungu bemisipha, ukudideka, kwaphinde kwaba nokungezwani kwezigodi yangaphakathi. Ezimweni ezingavamile, kukhona izinguquko ebuntwini, izitho babe ingazweli, kukhona Ukudlikizela futhi babone izinto ezingekho.
Ngemva kokumisa ukwelashwa resumption okungenzeka ukuqwasha lezivakashi neqembu elilodwa izimpawu lokuhoxa. Ngakho-ke, ukuqedela yokwelapha kumele kube kancane kancane.
Uma emva kokwelashwa "Somnolom" asesenenkinga ngilale noma uvuka ebusuku ukukhathazeka ukugwema ukubonakala ukulahlekelwa amandla okukhumbula anterograde, okuyiluthayo Kunconywa ukuthatha nje ngaphambi sokulala.
Sebenzisa ngesikhathi sokukhulelwa
Ukuntuleka kokukhulumisana nobufakazi basemtholampilo - isizathu esikhulu wamenza wenqaba "Somnola" engxenyeni yezinyanga ezintathu zokuqala zokukhulelwa. Uma kudingekile, avunyelwe ukusebenzisa izidakamizwa ezinyangeni zokugcina bephethe ingane, kodwa kuphela ngemithamo omncane.
Zopiclone, oyingxenye ye "Somnola" engxenyeni yezinyanga ezintathu 3rd sokukhulelwa kungabangela ukukhubazeka okukhulu izimpawu umbungu ka hypothermia kanye hypotension, kufanele kuphawulwe amathuba ukucindezeleka zokuphefumula futhi ukozela ngokweqile. Usana ezinsukwini zokuqala zokuphila kungenzeka wawubonakalisa lokuhoxa syndrome.
Uma izidakamizwa kunikezwa abesifazane yokuzala, kufanele siqaphele isidingo uthintane kuchwepheshe ukuze isinqumo ukuqedwa ukwelashwa uma kwenzeka uhlela ukukhulelwa.
Njengoba ketshezi asebenzayo "Somnola" excreted ku ubisi lwebele, umuthi phakathi ibele kungabangela ukubukeka ngobuthakathaka kwehle ithoni ngayo lapho usana.
Ukugcinwa Kwazo Ngenjongo iholide Pharmacy
Gcina elele izidakamizwa isidingo ome, nalapho kufinyelela khona izingane, lapho ingaziwa khona elangeni ngqo futhi lapho izinga lokushisa ingeqi degrees 25.
Thenga imithi kungaba yisilinganiso sesifundo ruble 200, futhi kuphela uma kukhona somuthi nokusetshenziswa kwawo sikadokotela, it is ayenzelwanga ukusetshenziswa ezizimele.
Izidakamizwa "Somnol": yokusetshenziswa, analogs
Uphenyo okuyiluthayo eziphikisa. Abanye bathi uma uthatha izidakamizwa, bakwazi ukuqeda ukuqwasha, ikhanda kanye njalo awakenings nasebusuku. Ezinye iziguli ukuthola ukuthi izidakamizwa ayikhululwa kubo kusukela izinkinga ezikhona.
Kunoma yikuphi, uma umuthi ezithathwe iseluleko sikadokotela, okulandelayo ngokucacile imiyalelo kahle ukuze abhekane nokuhlukaniswa ukuqwasha izidakamizwa "Somnol". Analogs, izinkomba yayo engase yehluke, asikho isenzo ayisasebenzi. Izidakamizwa aziwa kakhulu ase-izenzo ezifanayo zihlanganisa:
- "Sonovan";
- "Imovan";
- "Andante";
- "Selofen";
- "Zopiclone";
- "Adorma";
- "Normason";
- "Sonata";
- "Donormil";
- "Piklon".
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