Umuthi 'Spitomin ": yokusetshenziswa, izimpawu, contraindications

Namhlanje ukunitshela ngaloNkulunkulu izidakamizwa eziyingozi, njengezinto "Spitomin". Yokusetshenziswa, intengo, ukubuyekezwa, analogs kanye nezici zayo - zonke lezi zikhathi iziguli nesithakazelo ukuthi udokotela uye ebekiwe lokhu imithi. Lonke ulwazi oludingekayo zingatholakala kamuva kulesi sihloko.

Incazelo izidakamizwa, ezakheke, kanye nokwakheka emaphaketheni

Uyini izidakamizwa "Spitomin"? Yokusetshenziswa (ukulungiselela echazwe kulo mBhalo uvezwa ngemininingwane okukhulu) uveza ukuthi leli philisi ayinaphunga ezimhlophe, ukuma isiyingi futhi flat, nge chamfer kanye Valium futhi oqoshiwe «E151».

Ithuluzi iqukethe hydrochloride buspirone futhi izingxenye asizayo ezifana isitashi carboxymethyl, monohydrate lactose, magnesium stearate, sodium, microcrystalline cellulose futhi colloidal Silica anhydrous.

Ngo ukudayiswa izidakamizwa iza ibhamuza amaphakethe kanye amabhokisi.

Umgomo we operation

Iziphi izici ziyatholakala izidakamizwa "Spitomin"? Yokusetshenziswa (amaphilisi intengo abekwe ngezansi) uveza ukuthi lesi ejenti anxiolytic, esiphathelene uchungechunge non-benzodiazepine futhi ine umphumela antidepressant.

Ngokungafani nezinye anxiolytics, lokhu izidakamizwa abuzange antiepileptic, sine okuyiluthayo futhi izakhiwo myorelaxant. isimiso sayo wokusebenza kusekelwe imithelela buspirone ku dopaminergic futhi serotonergic izinhlelo.

Lokhu kusho ngokukhetha ekuvimbeni receptor Dopamine (presynaptic) futhi kwandisa izinga excitation izinzwa (Dopamine) ubuchopho obuphakathi.

Yini izakhiwo nezinye esivela izidakamizwa "Spitomin"? Yokusetshenziswa uthi Buspirone kuyinto agonist abakhethayo olulinganiselwe 5-HT1A serotonin receptor. It akuphazamisi yokubopha benzodiazepine receptor neGabha ibingamakhulu amathandathu, futhi akuphazamisi lengqondo umsebenzi futhi akabubangeli ukubekezelelana. Ngaphezu kwalokho, leli thuluzi akusho potentiate umphumela iziphuzo ezidakayo.

Umthelela zokwelapha zomuthi kubhekwe eba kancane kancane futhi kwenzeka emva elilodwa noma amabili ngemva kokwelashwa.

Kinetics kwezimali

Absorption zomuthi "Spitomin", yokusetshenziswa oboniswe ngezansi, kwenzeka pheshana emathunjini. Buspirone lisasetshenziswa akheka phakathi nokuwela kwawo isibindi. bioavailability Its 4% kanye esiphezulu plasma lokuhlushwa kufinyelelwe ngemva kwehora elilodwa.

Buspirone ikhishwe kanye ubisi. Ukuze uthole ulwazi mayelana Ukungena zomuthi ngokusebenzisa isithiyo esinomhlapho entulekayo.

Ukulungiselela ethathwe indle amahora amahlanu.

ubufakazi

Kusukela lokho okunqunyiwe "Spitomin" ithebhulethi? Yokusetshenziswa ukhombise izinkomba ezilandelayo:

• autonomic ukungasebenzi syndrome;
• abanenkinga yokukhathazeka kuyinto generalized;
• ukuhoxiswa syndrome utshwala (yokwelapha adjuvant);
• netwetwe disorder ;
• iziyaluyalu bacindezeleke (yokwelapha adjuvant).

Izimo

Kwezinye izimo, it is hhayi Kunconywa ukusebenzisa amaphilisi "Spitomin"? Yokusetshenziswa ithi pathologies elandelayo nemibandela umthamo imithi contraindicated ngaphansi lapho:

• ukufiphala;
• hypersensitivity kuya izithako zomuthi;
• myasthenia gravis;
• esingamahlalakhona kwezinso, ezinzima;
• yobudala ezincane;
• reception ngesikhathi esisodwa mao inhibitor ;
• lactation;
• ngesikhathi sokukhulelwa.

Nge-ejenti ukunakekelwa iqondiswa e isibindi sibe sesomile futhi ukwehluleka kwezinso.

Nomuthi "Spitomin": yokusetshenziswa

Analogs zomuthi izokwethulwa ngezansi.

Kulaba izimali okumele zithathwe esifanayo sosuku, ngaphambi noma ngemva kokudla.

Umuthi asivunyelwe ukusebenzisa ngezikhathi ezithile (ngokufunwa) ukwelapha ukukhathazeka, njengoba umphumela zayo zokwelapha eba ukusetshenziswa kuphela ngemva okuphindaphindiwe.

Umthamo le imithi ikhethwa ngamunye. Imvama, kuba 15 mg. Kufanele kube izingxenye 2-3 Ukweqiwa.

esiphezulu I umthamo owodwa kuyinto 30 mg kanye sangemihla - 60 mg.

Kwasebekhulile kwenziwa ushintsho of umthamo liyadingeka. Lapho kahle nomuthi kwezinso noma hepatic kumele kusetshenziswe ngokuqapha ngemithamo emincane.

side effects

Ngokuvamile imithi "Spitomin 'ebekezelele ngokubhekakade kahle. Kuphela kwezinye izimo, leli thuluzi ukwephulwa ezithile:

• ubuhlungu besifuba, unenkinga, yokufikelwa, isiyezi, hypotension, ikhanda, umfutho ophakeme wegazi,
• ukukhathazeka sezinzwa, cerebral iziyaluyalu kwegazi, ukusabela dysphoric, decompensation ephethwe yisifo senhliziyo, ukuzwela anda ukuze umsindo, isilethikusebenza, dysphoria, zenhliziyo, ecabanga ukuzibulala bradycardia;
• depersonalization, ukungabekezelelani abandayo, bajabula, claustrophobia, hyperkinesis, tinnitus, ukukhathazeka, ukulunywa emehlweni, ukucobeka, iso ububomvu, ukuhhema, amalimi awahlobene nalokho, ukudideka, iziyaluyalu ingqondo;
• angaboni kahle, laryngitis, conjunctivitis, ukuvuvukala mucosa acinene, ukunambitheka kahle, umuzwa wobukhulu esifubeni, endlebeni neziyaluyalu, hyperventilation, ubuhlungu iso, ukuntuleka komoya, photophobia, epistaxis, waqinisa intraocular;
• galaktoreyu, isicanucanu, umonakalo yegilo, ukubuyisa, enuresis ebusuku, sokuzincisha, isifiso ukwanda, dysuria, amathe, iziyaluyalu kokuya esikhathini, ukopha emathunjini, ejaculation imisiwe nezinye.

Inani, analogue, ukubuyekezwa

Izindleko zalesi ejenti kuyinto ruble angu-600. Uma kudingeka, lokhu kufakwa analog ezifana "Buspirone Sandoz."

Izibuyekezo Umthengi wazise ukuthi izidakamizwa okukhulunywa eyisidalwa esinenkululeko ezinhle anxiolytic. Nokho, kungase kuthathe kuphela onguchwepheshe ngenhloso isikhathi eside (hhayi ngezikhathi ezithile).