ImpiloAmalungiselelo

"Neuromidin": isitatimende

The main isithako zomuthi "Neuromidin" imfundo libizwa ukuxuba eziyinkimbinkimbi - ipidacrine. Amandla ayo kwemithi ngenxa inhlanganisela imiphumela ezimbili ezenzeka ezingeni yamangqamuzana ezinto eziphilayo. Eyokuqala wabo - ikhono ukwakha ukuvinjelwa potassium permeability we ulwelwesi, kanti eyesibili - kungenzeka okusithiyayo womsebenzi cholinesterase. Ngenxa ukubonakaliswa miphumela, lesi sidakamizwa "Neuromidin" sithuthukisa isenzo ejenti ezifana epinephrine, serotonin futhi histamine ku bushelelezi imisipha acetylcholine.

Umuthi usenamakhono elandelayo kwemithi. Kungaba zishukumisa ngempumelelo izinqubo yokudlulisela kwamanyuroni, futhi neqhaza ekulinganiseni ishayela at azungeze isimiso sezinzwa. Ukusebenzisa izidakamizwa ithuthukisa contractility ka bushelelezi imisipha izitho, futhi ngaphezu kwalokho, inikeza ukushukuma lolingene CNS.

Umuthi iphephile ngokwanele uma kusetshenziselwa kuhambisana nemibandela Kunconywa, ke akunamthelela teratogenic futhi mutagenic zomuthi akuyona isinyathelo umdlavuza futhi immunotoxic. Igalelo eyaba nalo omubi obuntu endocrine uhlelo kungukuthi uyalandelwa.

Ipidacrine uyakwazi ngokushesha angena ngemva kokuphathwa. Ngo esiphezulu plasma lokuhlushwa yayo kufinyelelwe emva ihora elilodwa esimweni uma imithi sathathwa ngesimo amaphilisi. Ukube ubukhona umuthi iqondiswa intramuscularly, emakamu esiphezulu kufinyelelwe ngesigamu isikhathi. Ekulungiseleleni plasma izicubu ngakho ngokushesha kuziwa ukuthi izinsalela kwakhona% 2 kuphela. Ipidacrine isigamu-ukuphila imizuzu 40, degree of ebudlelwaneni bayo nalowo amaprotheni kulingana 40-50%. Umuthi 'Neuromidin "manual uncoma ukusebenzisa izimo ezilandelayo. Kuyinto ikhambi eliphumelelayo ahlukahlukene izilonda isimiso sezinzwa. Ikakhulukazi, isetshenziswa ekwelapheni peripheral, izinhlobo ezahlukene neuritis, bulbar ukukhubazeka, inkumbulo iziyaluyalu.

Linqume izidakamizwa iziguli Alzheimer futhi izinhlobo ezahlukene komqondo, kanye amacala CNS izilonda imisuka ehlukahlukene. Medicine "Neuromidin" isetshenziswa ekwelashweni eziyinkimbinkimbi ekwelapheni CNS izifo demielinizuyuschih.

Ngaphambi kokusebenzisa izidakamizwa kufanele uzifunde ngokucophelela ukuze imiyalelo Kunconywa ukusetshenziswa kwezidakamizwa "Neuromidin" e amaphilisi kanye amaphilisi. Lesi sidingo ngokwengxenye kungenxa yokuthi i-ejenti senzelwe ekwelapheni ibanga ngokwanele ezibanzi izifo, futhi esimweni ngasinye indlela ngamunye, kokubili uhlobo abaphathi, kanye umthamo.

ukwelashwa Pi nale izidakamizwa kufanele uqaphele ukuthi kukhona contra-izinkomba, okuyiwona imithi Kunconywa. I Izimo eziyinhloko zihlanganisa isifo sokuwa, angina, ezahlukene wamathumbu isifo. Kufanele wokudeda abesifazane abakhulelwe kanye nalabo lapho kukhona hypersensitivity kuya izingxenye izidakamizwa.

Ngo ukwelashwa izidakamizwa, "Neuromidin" imfundo sinika kungenzeka inombolo yemiphumela emibi: ukulunywa, ukuqubuka, isicanucanu, isiyezi. Uma izenzakalo ezinjalo zenzeka, udinga ukwehlisa isilinganiso semithi oyidlayo noma ume isikhashana ukuthatha izidakamizwa.

ngokuqapha ikakhulukazi lapho ithola imithi ukuze babonwe yalezo ziguli uxilongwe izifo zenhliziyo.

Asincomi ngokuthatha izidakamizwa ngenkathi ushayela.

Nge ukweqisa izidakamizwa zomuthi ingxenye "Neuromidin" manual lichaza izimpawu ezifana bronchospasm, amehlo zamanzi. Kukhona futhi amacala myositis, ka ukuhlanza, futhi arrhythmias. Emacaleni angu-olunzima, kungase kube Ukudlikizela futhi equlekile kuqala.

Uma imithi ubuthi ingxenye kumele kusetshenziswe M-holinoblokatory: sulfate atropine, tsiklodol kanye nodokotela ngokushesha.

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